SCHEMBL4590917

SCHEMBL4590917

NC1CCCC(NC(=O)c2cccc(OC(F)(F)F)c2)CC1

nearest known ligand 0.59

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
TAS1R3 Q7RTX0 1/20 0.59
TAS1R1 Q7RTX1 1/20 0.59
TAS1R2 Q8TE23 1/20 0.59
SMYD3 Q9H7B4 7/20 0.56
PKM P14618 1/20 0.55
NPC1 O15118 1/20 0.54
HPGD P15428 1/20 0.52
RAB9A P51151 1/20 0.52
SMN1; SMN2 Q16637 1/20 0.52
MCHR1 Q99705 1/20 0.51
EPHX2 P34913 1/20 0.49
CCR2 P41597 1/20 0.49
PRSS1 P07477 2/20 0.49
PRSS2 P07478 2/20 0.49
PRSS3 P35030 2/20 0.49
ST14 Q9Y5Y6 2/20 0.49
F2 P00734 1/20 0.48
GRM5 P41594 2/20 0.48
KDM1A O60341 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2472926 0.89 TAS1R3 (0.67) TAS1R3TAS1R1TAS1R2SMYD3PKM
SCHEMBL4609353 0.84 TAS1R3 (0.62) TAS1R3TAS1R1TAS1R2PKMNPC1
SCHEMBL4575139 0.81 TAS1R3 (0.61) TAS1R3TAS1R1TAS1R2PKMNPC1
SCHEMBL6455818 0.80 SMYD3 (0.58) SMYD3MCHR1EPHX2PRSS1PRSS2
SCHEMBL6455822 0.80 SMYD3 (0.58) SMYD3MCHR1EPHX2PRSS1PRSS2
SCHEMBL6455626 0.79 SMYD3 (0.69) SMYD3PKMNPC1HPGDRAB9A
SCHEMBL6455623 0.79 SMYD3 (0.69) SMYD3PKMNPC1HPGDRAB9A
SCHEMBL1580017 0.77 TAS1R3 (0.58) TAS1R3TAS1R1TAS1R2PKMNPC1
SCHEMBL10294731 0.76 NPC1 (0.66) TAS1R3TAS1R1TAS1R2SMYD3PKM
SCHEMBL4574282 0.75 USP30 (0.60) TAS1R3TAS1R1TAS1R2PKMHPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008065500-A2 HETEROARYL AMIDES AS TYPE I GLYCINE TRANSPORT INHIBITORS PFIZER PRODUCTS INC. (US) 2008-06-05 WO disclosed