SCHEMBL4591279

SCHEMBL4591279

Cc1c[nH]c(-c2ccc(C(F)F)cc2C#N)n1

nearest known ligand 0.35

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
HSP90AB1 P08238 6/20 0.35
ROCK2 O75116 1/20 0.33
ROCK1 Q13464 1/20 0.33
JAK2 O60674 1/20 0.33
JAK3 P52333 1/20 0.33
LIMK1 P53667 1/20 0.33
LIMK2 P53671 1/20 0.33
MCL1 Q07820 1/20 0.33
CYP11B1 P15538 2/20 0.32
CYP11B2 P19099 2/20 0.32
TRPA1 O75762 1/20 0.31
GRM5 P41594 1/20 0.31
KDM5A P29375 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4590957 0.83 HSP90AB1 (0.45) HSP90AB1JAK2JAK3LIMK1LIMK2
SCHEMBL4591503 0.81 HSP90AB1 (0.42) HSP90AB1MCL1CYP11B1CYP11B2
SCHEMBL2323777 0.79 PTGES (0.38) HSP90AB1MCL1KDM5A
SCHEMBL4590941 0.79 MCL1 (0.39) HSP90AB1MCL1KDM5A
SCHEMBL4591479 0.79 HSP90AB1 (0.34) HSP90AB1CYP11B1CYP11B2TRPA1KDM5A
SCHEMBL3633331 0.79 KDM4E (0.41) HSP90AB1MCL1
SCHEMBL4591744 0.78 XDH (0.40) HSP90AB1TRPA1
SCHEMBL4592503 0.77 PDE4B (0.42) HSP90AB1
SCHEMBL4591549 0.75 DHODH (0.41) HSP90AB1TRPA1KDM5A
SCHEMBL4592321 0.75 TRPA1 (0.42) TRPA1GRM5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1937688-A1 IMIDAZO BENZODIAZEPINE DERIVATIVES F.HOFFMANN-LA ROCHE AG (CH) 2008-07-02 EP disclosed
WO-2007042421-A1 IMIDAZO BENZODIAZEPINE DERIVATIVES F. HOFFMANN-LA ROCHE AG (CH) 2007-04-19 WO disclosed