SCHEMBL4591313

SCHEMBL4591313

CCOc1cc(C=O)ccc1-c1ncc[nH]1

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 9/20 0.52
TACR2 P21452 1/20 0.44
HPGD P15428 2/20 0.41
TDP1 Q9NUW8 2/20 0.41
L3MBTL1 Q9Y468 2/20 0.41
MAPT P10636 2/20 0.41
NPSR1 Q6W5P4 1/20 0.41
KDM4E B2RXH2 3/20 0.41
FDPS P14324 1/20 0.40
DHFR P00374 1/20 0.39
TSHR P16473 1/20 0.38
VCP P55072 1/20 0.38
RXFP1 Q9HBX9 1/20 0.38
CYP1A2 P05177 1/20 0.38
CYP3A4 P08684 1/20 0.38
CYP2D6 P10635 1/20 0.38
CYP19A1 P11511 1/20 0.38
CYP2C9 P11712 1/20 0.38
CYP2C19 P33261 1/20 0.38
GAA P10253 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4591361 0.83 ALDH1A1 (0.44) ALDH1A1TACR2HPGDTDP1L3MBTL1
SCHEMBL2960690 0.77 ALDH1A1 (0.55) ALDH1A1TACR2HPGDTDP1L3MBTL1
SCHEMBL12087983 0.77 VCP (0.38) DHFRVCPCYP1A2CYP3A4CYP2D6
SCHEMBL3403159 0.76 ADRA1A (0.58) ALDH1A1HPGDNPSR1KDM4EVCP
SCHEMBL18519805 0.75 ALDH1A1 (0.47) ALDH1A1MAPTKDM4ECYP1A2CYP3A4
SCHEMBL2599782 0.74 ALDH1A1 (0.51) ALDH1A1TACR2HPGDTDP1L3MBTL1
SCHEMBL17535846 0.74 ALDH1A1 (0.58) ALDH1A1TACR2HPGDTDP1L3MBTL1
SCHEMBL2955584 0.74 ALDH1A1 (0.58) ALDH1A1TACR2HPGDTDP1L3MBTL1
SCHEMBL493684 0.73 ALDH1A1 (0.73) ALDH1A1TACR2HPGDTDP1L3MBTL1
SCHEMBL30159697 0.73 ALDH1A1 (0.73) ALDH1A1TACR2HPGDTDP1L3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1893603-A1 PIPERIDIN-4-YL-AMIDE DERIVATIVES AND THEIR USE AS SST RECEPTOR SUBTYPE 5 ANTAGONISTS F. Hoffmann-La Roche AG (CH) 2008-03-05 EP disclosed
WO-2006128803-A1 PIPERIDIN-4-YL-AMIDE DERIVATIVES AND THEIR USE AS SST RECEPTOR SUBTYPE 5 ANTAGONISTS F. HOFFMANN-LA ROCHE AG (CH) 2006-12-07 WO disclosed