SCHEMBL4592387

SCHEMBL4592387

CCc1ccc(N)c(CC)c1NC(=O)N(CC1CCCCC1)c1ccc(C(C)C)cc1.CCc1ccc(N)c(CC)c1NC(=O)N(Cc1ccc(OC)cc1F)c1ccc(C(C)C)cc1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CTSD P07339 2/20 0.37
C5AR1 P21730 2/20 0.36
GPR183 P32249 1/20 0.35
ADGRF1 Q5T601 1/20 0.35
GPR65 Q8IYL9 1/20 0.35
PSEN1 P49768 1/20 0.33
PSEN2 P49810 1/20 0.33
APH1B Q8WW43 1/20 0.33
NCSTN Q92542 1/20 0.33
APH1A Q96BI3 1/20 0.33
PSENEN Q9NZ42 1/20 0.33
HDAC3 O15379 1/20 0.33
HDAC1 Q13547 1/20 0.33
HDAC2 Q92769 1/20 0.33
HDAC8 Q9BY41 1/20 0.33
HDAC6 Q9UBN7 1/20 0.33
HTR2A P28223 1/20 0.33
ALDH1A1 P00352 1/20 0.32
PTK2 Q05397 1/20 0.32
MEN1 O00255 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4591774 0.95 CTSD (0.34) CTSDC5AR1GPR183ADGRF1GPR65
SCHEMBL4592692 0.91 PTK2 (0.37) C5AR1GPR183ADGRF1GPR65HTR2A
SCHEMBL4592545 0.87 EPHX1 (0.40) L3MBTL1
SCHEMBL4591758 0.85 RORC (0.34) CTSDC5AR1GPR183ADGRF1GPR65
SCHEMBL4592456 0.82 PTK2 (0.35) C5AR1GPR183ADGRF1GPR65PTK2
SCHEMBL12047724 0.82 ALDH1A1 (0.40) C5AR1GPR183ADGRF1GPR65ALDH1A1
SCHEMBL4592440 0.79 BCL2A1 (0.40) C5AR1GPR183ADGRF1GPR65ALDH1A1
SCHEMBL4592857 0.77 EPHX1 (0.39)
SCHEMBL4592636 0.76 KDM4E (0.32) ALDH1A1PTK2MEN1POLBKMT2A
SCHEMBL4592639 0.76 KDM4E (0.32) ALDH1A1PTK2MEN1POLBKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1885691-A1 C5A RECEPTOR ANTAGONISTS Jerini AG (DE) 2008-02-13 EP disclosed
WO-2006128670-A1 C5A RECEPTOR ANTAGONISTS JERINI AG (DE) 2006-12-07 WO disclosed