SCHEMBL4592679

SCHEMBL4592679

CCc1c(N)cc(Cl)c(CC)c1NC(=O)N(Cc1ccc(C(F)(F)F)cc1)c1ccc(C(C)C)cc1.CCc1ccc(N)c(CC)c1NC(=O)N(Cc1ccc(OC)nc1)c1ccc(C(C)C)cc1

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
OXTR P30559 1/20 0.35
NR3C1 P04150 1/20 0.33
CETP P11597 5/20 0.33
LMNA P02545 2/20 0.33
GAA P10253 1/20 0.33
NPSR1 Q6W5P4 1/20 0.33
PDK1 Q15118 1/20 0.32
GCGR P47871 2/20 0.32
GIPR P48546 2/20 0.32
PRKAB2 O43741 1/20 0.32
PRKAG1 P54619 1/20 0.32
PRKAA2 P54646 1/20 0.32
PRKAA1 Q13131 1/20 0.32
PRKAG3 Q9UGI9 1/20 0.32
PRKAG2 Q9UGJ0 1/20 0.32
PRKAB1 Q9Y478 1/20 0.32
OPRM1 P35372 1/20 0.32
KCNH2 Q12809 1/20 0.31
MCHR1 Q99705 1/20 0.31
PDK2 Q15119 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4592247 0.89 OXTR (0.42) OXTRLMNAGAANPSR1
SCHEMBL4592839 0.88 OXTR (0.44) OXTR
SCHEMBL4592643 0.86 PDK1 (0.40) CETPLMNAPDK1GCGRGIPR
SCHEMBL4591943 0.85 PDK2 (0.38) CETPLMNAPDK1GCGRGIPR
SCHEMBL4592189 0.83 C5AR1 (0.37) PDK1
SCHEMBL4592072 0.83 KCNH2 (0.37) NPSR1KCNH2
SCHEMBL4592810 0.81 UTS2R (0.35) CETPPDK1PDK2PDK4
SCHEMBL4592138 0.81 CNR2 (0.34) LMNAPDK1
SCHEMBL4592388 0.80 MAPT (0.38) LMNAPDK1
SCHEMBL4591539 0.80 LMNA (0.34) LMNAPDK1PDK2PDK4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1885691-A1 C5A RECEPTOR ANTAGONISTS Jerini AG (DE) 2008-02-13 EP claimed
WO-2006128670-A1 C5A RECEPTOR ANTAGONISTS JERINI AG (DE) 2006-12-07 WO claimed