SCHEMBL4592681

SCHEMBL4592681

O=C(N[C@@H](COC(I)c1ccccc1)CS(=O)(=O)Cl)OCc1ccccc1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CTRB1 P17538 2/20 0.47
ALDH1A1 P00352 6/20 0.42
CYP1A2 P05177 4/20 0.42
CTSL P07711 1/20 0.42
CTSS P25774 1/20 0.42
CA12 O43570 2/20 0.41
CA1 P00915 2/20 0.41
CA2 P00918 2/20 0.41
CA9 Q16790 2/20 0.41
CYP3A4 P08684 7/20 0.41
TSHR P16473 7/20 0.41
CASP1 P29466 2/20 0.41
SMN1; SMN2 Q16637 2/20 0.41
SYK P43405 1/20 0.41
ATM Q13315 1/20 0.41
CYP2C9 P11712 6/20 0.41
CYP2C19 P33261 5/20 0.41
LMNA P02545 2/20 0.41
MEN1 O00255 2/20 0.41
KMT2A Q03164 2/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL223417 0.83 CTRB1 (0.53) CTRB1CTSLCTSSCA12CA1
SCHEMBL11283166 0.81 CTRB1 (0.56) CTRB1ALDH1A1CA12CA1CA2
SCHEMBL18576677 0.81 CTRB1 (0.67) CTRB1ALDH1A1CTSLCTSSCA12
SCHEMBL2353282 0.81 CTRB1 (0.67) CTRB1ALDH1A1CTSLCTSSCA12
SCHEMBL31089911 0.74 CA2 (0.54) CTRB1CTSLCTSSCA12CA1
SCHEMBL2749553 0.74 PPARA (0.53) CTRB1CTSLCTSSCA12CA1
SCHEMBL30629995 0.74 CA2 (0.54) CTRB1CTSLCTSSCA12CA1
SCHEMBL2102910 0.74 CASP1 (0.52) CTRB1ALDH1A1CTSLCTSSCA12
SCHEMBL19136379 0.74 CA2 (0.54) CTRB1CTSLCTSSCA12CA1
SCHEMBL5559459 0.74 CTRB1 (0.51) CTRB1ALDH1A1CTSLCTSSCA12

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1888567-A1 HETEROARYL-CARBOXYLIC ACID (SULFAMOYL ALKYL) AMIDE - DERIVATIVES AS FACTOR XA INHIBITORS Sanofi-Aventis (FR) 2008-02-20 EP disclosed
WO-2006122661-A1 HETEROARYL-CARBOXYLIC ACID (SULFAMOYL ALKYL) AMIDE - DERIVATIVES AS FACTOR XA INHIBITORS SANOFI-AVENTIS (DE) 2006-11-23 WO disclosed