SCHEMBL4592925

SCHEMBL4592925

COc1c(CBr)cc(F)c(F)c1F

nearest known ligand 0.33

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 1/20 0.32
ALDH1A1 P00352 1/20 0.32
MEP1B Q16820 1/20 0.32
HTR2A P28223 1/20 0.30
HTR2C P28335 1/20 0.30
HTR2B P41595 1/20 0.30
TUBB1 Q9H4B7 1/20 0.30
CYP1A2 P05177 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3932880 0.84 MEP1B (0.35) MEP1BHTR2AHTR2CHTR2BTUBB1
SCHEMBL4592852 0.84 ALDH1A1 (0.35) ALDH1A1MEP1BHTR2AHTR2CHTR2B
SCHEMBL18543623 0.78 CYP1A2 (0.51) HTR2AHTR2CHTR2BCYP1A2
SCHEMBL29896365 0.76 MEP1B (0.41) ALDH1A1MEP1BHTR2AHTR2CHTR2B
SCHEMBL4592472 0.76 MEP1B (0.41) ALDH1A1MEP1BHTR2AHTR2CHTR2B
SCHEMBL3488489 0.76 ALDH1A1 (0.35) PTGS2ALDH1A1HTR2AHTR2CHTR2B
SCHEMBL3655636 0.74 MEP1B (0.35) ALDH1A1MEP1B
SCHEMBL6739577 0.73 TUBB1 (0.35) PTGS2ALDH1A1HTR2AHTR2CHTR2B
SCHEMBL826597 0.73 HDAC3 (0.33)
SCHEMBL4589673 0.72 CA2 (0.46) PTGS2TUBB1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1807398-B1 NEW INDOLE OR BENZIMIDAZOLE DERIVATIVES HOFFMANN LA ROCHE (CH) 2008-06-25 EP disclosed