SCHEMBL4592940

SCHEMBL4592940

CC(=O)NC1(C)CCN(Cc2ccc(Br)cc2)CC1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TNIK Q9UKE5 1/20 0.50
MMP1 P03956 2/20 0.48
MMP9 P14780 2/20 0.48
MMP13 P45452 2/20 0.48
ADAM17 P78536 2/20 0.48
POLB P06746 1/20 0.48
FAAH O00519 1/20 0.46
ALDH1A1 P00352 3/20 0.46
KDM4E B2RXH2 2/20 0.46
DRD2 P14416 1/20 0.46
GPR183 P32249 2/20 0.45
LMNA P02545 1/20 0.45
HPGD P15428 1/20 0.45
HTT P42858 1/20 0.45
MCHR1 Q99705 1/20 0.45
SIGMAR1 Q99720 1/20 0.44
NPC1 O15118 1/20 0.44
DPP4 P27487 1/20 0.44
MME P08473 1/20 0.44
CYP2D6 P10635 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1991966 0.86 CYP2D6 (0.59) POLBALDH1A1DRD2MCHR1SIGMAR1
Hydrochloric Acid SCHEMBL8416135 0.84 CYP2D6 (0.58) POLBALDH1A1KDM4EDRD2MCHR1
SCHEMBL24770881 0.78 MMP1 (0.54) TNIKMMP1MMP9MMP13ADAM17
SCHEMBL27042826 0.78 MMP1 (0.48) TNIKMMP1MMP9MMP13ADAM17
SCHEMBL17163855 0.78 CYP2D6 (0.53) ALDH1A1DRD2DPP4CYP2D6
SCHEMBL17082420 0.78 CYP2D6 (0.53) ALDH1A1DRD2DPP4CYP2D6
SCHEMBL953425 0.78 CYP2D6 (0.53) ALDH1A1DRD2DPP4CYP2D6
SCHEMBL4591580 0.77 ALDH1A1 (0.54) TNIKMMP1MMP9MMP13ADAM17
SCHEMBL1427542 0.77 ALDH1A1 (0.58) TNIKMMP1MMP9MMP13ADAM17
SCHEMBL32665256 0.76 ALDH1A1 (0.49) TNIKMMP1MMP9MMP13ADAM17

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-101296906-A (hetero)aryl compounds with MCH antagonistic activity and medicaments comprising these compounds BOEHRINGER INGELHEIM INT (DE) 2008-10-29 CN disclosed
EP-1943231-A1 (HETERO)ARYL COMPOUNDS WITH MCH ANTAGONISTIC ACTIVITY AND MEDICAMENTS COMPRISING THESE COMPOUNDS BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2008-07-16 EP disclosed
US-20070111981-A1 New (hetero)aryl compounds with MCH antagonistic activity and medicaments comprising these compounds ROTH GERALD J 2007-05-17 US disclosed
WO-2007048802-A1 (HETERO)ARYL COMPOUNDS WITH MCH ANTAGONISTIC ACTIVITY AND MEDICAMENTS COMPRISING THESE COMPOUNDS BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2007-05-03 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20070111981-A1 New (hetero)aryl compounds with MCH antagonistic activity and medicaments comprising these compounds MCHR1, GPR119, MCHR2 TNIK 4757/4885MMP1 4859/4885MMP9 4867/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.