SCHEMBL4592970

SCHEMBL4592970

O=C(O)NC(CCS(=O)(=O)Cl)C(=O)OCc1ccccc1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TACR1 P25103 1/20 0.44
ALDH1A1 P00352 3/20 0.44
CA12 O43570 2/20 0.43
CA1 P00915 2/20 0.43
CA2 P00918 2/20 0.43
CA9 Q16790 2/20 0.43
POLB P06746 1/20 0.43
CASP1 P29466 3/20 0.41
ACE P12821 1/20 0.41
LMNA P02545 1/20 0.40
MBTPS1 Q14703 1/20 0.40
CTSL P07711 1/20 0.40
CTSS P25774 1/20 0.40
CTRB1 P17538 2/20 0.40
CTSK P43235 1/20 0.40
MAPK1 P28482 1/20 0.40
L3MBTL1 Q9Y468 1/20 0.40
SLC6A2 P23975 1/20 0.40
SLC6A3 Q01959 1/20 0.40
KMT2A Q03164 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30788894 0.91 CASP1 (0.51) TACR1ALDH1A1CA12CA1CA2
SCHEMBL1290959 0.86 CTSL (0.52) ALDH1A1CASP1CTSLCTSSCTSK
SCHEMBL1290957 0.86 CTSL (0.52) ALDH1A1CASP1CTSLCTSSCTSK
SCHEMBL8346395 0.83 SIRT2 (0.52) TACR1CASP1CTSLCTSSCTSK
SCHEMBL4212334 0.81 TACR1 (0.49) TACR1ALDH1A1POLBACEMBTPS1
SCHEMBL7598622 0.79 TACR1 (0.47) TACR1ALDH1A1CA12CA1CA2
SCHEMBL24111516 0.78 TACR1 (0.66) TACR1ALDH1A1POLBACEMBTPS1
SCHEMBL2102910 0.77 CASP1 (0.52) TACR1ALDH1A1CA12CA1CA2
SCHEMBL28709501 0.76 ALDH1A1 (0.53) TACR1ALDH1A1POLBCASP1ACE
SCHEMBL11432342 0.74 CTSK (0.61) ALDH1A1CTSLCTSSCTSKKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1888567-A1 HETEROARYL-CARBOXYLIC ACID (SULFAMOYL ALKYL) AMIDE - DERIVATIVES AS FACTOR XA INHIBITORS Sanofi-Aventis (FR) 2008-02-20 EP disclosed
WO-2006122661-A1 HETEROARYL-CARBOXYLIC ACID (SULFAMOYL ALKYL) AMIDE - DERIVATIVES AS FACTOR XA INHIBITORS SANOFI-AVENTIS (DE) 2006-11-23 WO disclosed