SCHEMBL4593314

SCHEMBL4593314

O=COc1ccc(Cl)cc1Cl

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TTR P02766 3/20 0.49
TDP1 Q9NUW8 3/20 0.48
MAPT P10636 2/20 0.47
NR1I2 O75469 1/20 0.47
LMNA P02545 1/20 0.47
PGR P06401 1/20 0.47
HSP90AA1 P07900 1/20 0.47
ADORA3 P0DMS8 1/20 0.47
HSPA5 P11021 1/20 0.47
HPGD P15428 1/20 0.47
CBR1 P16152 1/20 0.47
TBXA2R P21731 1/20 0.47
SLC6A2 P23975 1/20 0.47
AGTR1 P30556 1/20 0.47
SLC6A3 Q01959 1/20 0.47
S1PR4 O95977 2/20 0.45
KMT2A Q03164 1/20 0.44
TP53 P04637 1/20 0.42
TSHR P16473 1/20 0.42
PLA2G1B P04054 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28746894 0.98 TTR (0.47) TTRTDP1MAPTNR1I2LMNA
SCHEMBL8665449 0.83 TDP1 (0.43) TTRTDP1MAPTLMNATP53
SCHEMBL11084246 0.79 TSHR (0.49) MAPTLMNAHPGDSLC6A2SLC6A3
SCHEMBL16546178 0.79 TTR (0.53) TTRTDP1MAPTNR1I2LMNA
SCHEMBL28086712 0.79 TTR (0.46) TTRTDP1MAPTNR1I2LMNA
SCHEMBL12121021 0.79 ACHE (0.43) TDP1MAPTLMNAHPGDS1PR4
SCHEMBL9775676 0.79 SLC6A2 (0.41) HPGDSLC6A2SLC6A3S1PR4KMT2A
SCHEMBL15834997 0.79 MAPT (0.57) TTRTDP1MAPTLMNAHPGD
SCHEMBL28832700 0.79 CYP3A4 (0.46) TDP1MAPTHPGDKMT2ATSHR
SCHEMBL27584712 0.79 SMN1; SMN2 (0.43) TDP1LMNAHPGDS1PR4KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 73 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2636669-B1 PYRAZOLE AMIDE COMPOUND AND USE THEREOF AS FUNGICIDE SINOCHEM CORP (CN) 2015-10-21 EP claimed
US-8614214-B2 Pyrazole amide compounds and uses thereof SINOCHEM CORPORATION (CN) 2013-12-24 US claimed
EP-2636669-A1 PYRAZOLE AMIDE COMPOUND AND USE THEREOF Sinochem Corporation (CN) 2013-09-11 EP claimed
US-20130225585-A1 PYRAZOLE AMIDE COMPOUNDS AND USES THEREOF SHENYANG RESEARCH INSTITUTE OF CHEMICAL INDUSTRY CO., LTD. (CN) 2013-08-29 US claimed
CN-101014585-A Radically polymerizable sulfur-containing compound and radically polymerizable sulfur-containing polymer SHOWA DENKO KK (JP) 2007-08-08 CN claimed
CN-1976967-A Carboxylic acid modified aminoplast crosslinking agent and powder coating compositions PPG IND OHIO INC (US) 2007-06-06 CN claimed
EP-0354297-B1 THIADIAZINES, PROCESS FOR PRODUCTION THEREOF, AND INSECTICIDAL AND ACARICIDAL AGENTS COMPRISING THE THIADIAZINES MITSUI TOATSU CHEMICALS, Inc. (JP) 1992-08-05 EP claimed
US-5021412-A Protecting agricultural crops MITSUI TOATSU CHEMICALS, INC. (JP) 1991-06-04 US claimed
US-4537720-A N-substituted-2-(R)-(sulfinic acid)-3-(S)-(acylamino)-4-oxo-azetidines and process ELI LILLY AND COMPANY (US) 1985-08-27 US claimed
CN-112384511-B Endoparasite depsipeptides 硕腾服务有限责任公司 2024-01-30 CN disclosed
CN-113631548-B Serotonin 5-HT2B inhibiting compounds 硕腾服务有限责任公司 2023-06-06 CN disclosed
CN-108947804-A A kind of preparation method of chlorobenzene oxycarboxylic acid substance 山东润博生物科技有限公司 2018-12-07 CN disclosed
CN-108947803-A A kind of preparation method of phenoxy carboxylic acid substance 山东润博生物科技有限公司 2018-12-07 CN disclosed
CN-104341316-B Aryl amide derivative of one class two and preparation method thereof, pharmaceutical composition and purposes 中国科学院上海药物研究所 2017-07-28 CN disclosed
EP-0019760-B1 ESTERS OF 3-ARYL-5-METHYL-PYRAZOLE-4-CARBOXYLIC ACID, HERBICIDES CONTAINING THEM, PROCESS FOR THEIR PREPARATION AND THEIR USE BASF Aktiengesellschaft (DE) 1982-06-23 EP disclosed
US-4264495-A EXHIBITING GOOD COLOFASTNESS AND DYEABILITY ON POLYAMIDES AND OTHER FIBERS EASTMAN KODAK COMPANY (US) 1981-04-28 US disclosed
US-4259350-A PROTECTING DEGRADABLE ORGANIC MATERIAL FROM FUNGAL OR INSECT ATTACK SANKYO COMPANY LIMITED (JP) 1981-03-31 US disclosed
EP-0019760-A1 Esters of 3-aryl-5-methyl-pyrazole-4-carboxylic acid, herbicides containing them, process for their preparation and their use BASF Aktiengesellschaft (DE) 1980-12-10 EP disclosed
US-4070352-A COLORFAST, SUBLIMATION AND OZONE RESISTANT BLUE AZO DYES FOR POLYAMIDES EASTMAN KODAK COMPANY (US) 1978-01-24 US disclosed
US-3932419-A QUINOLINE DYES BAYER AKTIENGESELLSCHAFT (DT) 1976-01-13 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20130225585-A1 PYRAZOLE AMIDE COMPOUNDS AND USES THEREOF BROX, OAT, CAT TTR 2960/4885TDP1 4236/4885MAPT 288/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.