SCHEMBL4593659

SCHEMBL4593659

N=C(N)c1cccc(S(N)(=O)=O)c1O

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CDK2 P24941 1/20 0.47
CA1 P00915 9/20 0.44
CA2 P00918 9/20 0.44
CA9 Q16790 7/20 0.44
CA5A P35218 3/20 0.42
STAT3 P40763 1/20 0.42
MAPK1 P28482 1/20 0.40
CA6 P23280 3/20 0.39
CA12 O43570 3/20 0.39
CA4 P22748 2/20 0.39
CYP2C9 P11712 2/20 0.39
CA7 P43166 2/20 0.39
CA5B Q9Y2D0 2/20 0.39
CA14 Q9ULX7 1/20 0.39
MCL1 Q07820 1/20 0.39
HSD17B10 Q99714 1/20 0.39
F10 P00742 3/20 0.39
PRSS1 P07477 2/20 0.39
PRSS2 P07478 2/20 0.39
PRSS3 P35030 2/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4593438 0.82 CA1 (0.56) CDK2CA1CA2CA9CA5A
SCHEMBL3559324 0.76 ALDH1A1 (0.50) CDK2CA1CA2MAPK1CA6
SCHEMBL5518503 0.76 CDK2 (0.63) CDK2CA1CA2CA9CA5A
SCHEMBL1121320 0.72 CA1 (0.61) CDK2CA1CA2CA9CA5A
SCHEMBL8988809 0.72 GAA (0.38) CDK2CA1CA2CA9CA5A
SCHEMBL27523119 0.71 CA1 (0.51) CDK2CA1CA2CA9CA5A
SCHEMBL4658049 0.71 ALDH1A1 (0.52) CDK2CA1CA2CA9CA5A
SCHEMBL1685391 0.71 ALDH1A1 (0.52) CDK2CA1CA2CA9CA5A
SCHEMBL7562109 0.71 TTR (0.41) CA1CA2CA9CA5AF10
SCHEMBL6657862 0.71 CA1 (0.55) CDK2CA1CA2CA9CA5A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1934214-A1 OXADIAZOLYL PYRAZOLO-PYRIMIDINES AS MGLUR2 ANTAGONISTS F.HOFFMANN-LA ROCHE AG (CH) 2008-06-25 EP disclosed
WO-2007039439-A1 OXADIAZOLYL PYRAZOLO-PYRIMIDINES AS MGLUR2 ANTAGONISTS F.HOFFMANN-LA ROCHE AG (CH) 2007-04-12 WO disclosed