SCHEMBL4594394

SCHEMBL4594394

CCOc1cc(CN(c2nc3cc(C(=O)OC)ccc3s2)C2CCNCC2)cc(OCC)c1Cl

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SSTR1 P30872 1/20 0.39
SSTR5 P35346 1/20 0.39
TP53 P04637 2/20 0.35
MAPT P10636 3/20 0.35
LMNA P02545 1/20 0.35
SLC2A1 P11166 1/20 0.35
NPC1 O15118 3/20 0.34
RAB9A P51151 3/20 0.34
HSP90AA1 P07900 1/20 0.34
NR1H4 Q96RI1 1/20 0.34
TACR1 P25103 2/20 0.33
CREBBP Q92793 1/20 0.33
LIPG Q9Y5X9 1/20 0.33
KDM4E B2RXH2 1/20 0.33
KMT2A Q03164 1/20 0.33
SMN1; SMN2 Q16637 1/20 0.33
ALDH1A1 P00352 1/20 0.33
CNR2 P34972 1/20 0.33
HDAC6 Q9UBN7 1/20 0.33
PTK2 Q05397 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4593898 0.92 SSTR5 (0.45) SSTR1SSTR5TP53MAPTLMNA
SCHEMBL4593786 0.88 SSTR5 (0.35) SSTR5TP53MAPTLMNANPC1
SCHEMBL4593776 0.88 SSTR5 (0.40) SSTR1SSTR5HDAC6
SCHEMBL4593662 0.87 NPC1 (0.42) TP53MAPTNPC1RAB9AKDM4E
SCHEMBL4594269 0.85 SSTR5 (0.43) SSTR1SSTR5TP53MAPTNPC1
SCHEMBL4593460 0.82 SSTR5 (0.47) SSTR1SSTR5MAPTNPC1RAB9A
SCHEMBL4593487 0.82 TRPV1 (0.38) TP53MAPTNPC1RAB9AHSP90AA1
SCHEMBL4594733 0.82 TP53 (0.34) SSTR1SSTR5TP53MAPTLMNA
SCHEMBL4593912 0.81 SSTR5 (0.41) SSTR1SSTR5TP53MAPTLMNA
SCHEMBL4593554 0.80 SSTR5 (0.36) SSTR1SSTR5TP53MAPTLMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1924579-A2 BENZOOXAZOLE, OXAZOLOPYRIDINE, BENZOTHIAZOLE AND THIAZOLOPYRIDINE DERIVATIVES F.HOFFMANN-LA ROCHE AG (CH) 2008-05-28 EP claimed
WO-2007025897-A2 BENZOOXAZOLE, OXAZOLOPYRIDINE, BENZOTHIAZOLE AND THIAZOLOPYRIDINE DERIVATIVES F. HOFFMANN-LA ROCHE AG (CH) 2007-03-08 WO claimed
EP-1924579-A2 BENZOOXAZOLE, OXAZOLOPYRIDINE, BENZOTHIAZOLE AND THIAZOLOPYRIDINE DERIVATIVES F.HOFFMANN-LA ROCHE AG (CH) 2008-05-28 EP disclosed
WO-2007025897-A2 BENZOOXAZOLE, OXAZOLOPYRIDINE, BENZOTHIAZOLE AND THIAZOLOPYRIDINE DERIVATIVES F. HOFFMANN-LA ROCHE AG (CH) 2007-03-08 WO disclosed