SCHEMBL4595014

SCHEMBL4595014

CC(C)c1cc(CCCl)cc(C(C)C)c1O

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GSR P00390 1/20 0.55
GABRA1 P14867 6/20 0.54
GABRB1 P18505 5/20 0.54
GABRB2 P47870 4/20 0.53
GABRA5 P31644 2/20 0.53
GABRA3 P34903 2/20 0.53
GABRA2 P47869 2/20 0.53
GABRA4 P48169 2/20 0.53
GABRA6 Q16445 2/20 0.53
CA1 P00915 2/20 0.52
CA2 P00918 2/20 0.52
TRPA1 O75762 1/20 0.47
MAPT P10636 1/20 0.45
FAAH O00519 1/20 0.41
LMNA P02545 1/20 0.41
CYP1A2 P05177 1/20 0.41
CYP3A4 P08684 1/20 0.41
HPGD P15428 1/20 0.41
TSHR P16473 1/20 0.41
GABRG2 P18507 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6049696 0.83 GSR (0.59) GSRGABRA1GABRB1GABRB2GABRA5
SCHEMBL13057520 0.81 GSR (0.57) GSRGABRA1GABRB1GABRB2GABRA5
SCHEMBL4594369 0.79 GSR (0.55) GSRGABRA1GABRB1GABRB2GABRA5
SCHEMBL2467528 0.78 GSR (0.63) GSRGABRA1GABRB1GABRB2GABRA5
SCHEMBL11810825 0.78 GSR (0.53) GSRGABRA1GABRB1GABRB2GABRA5
SCHEMBL200138 0.78 GABRA1 (0.60) GSRGABRA1GABRB1GABRB2GABRA5
SCHEMBL6419829 0.78 GSR (0.53) GSRGABRA1GABRB1GABRB2GABRA5
SCHEMBL11519193 0.77 TRPA1 (0.52) GSRGABRA1GABRB1GABRB2GABRA5
SCHEMBL5692077 0.76 GABRA1 (0.54) GSRGABRA1GABRB1GABRB2GABRA5
SCHEMBL9193416 0.76 GABRA1 (0.54) GSRGABRA1GABRB1GABRB2GABRA5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4463187-A Process for the preparation of 3,5-dihydrocarbyl-4-hydroxybenzylmalonic acid esters ETHYL CORPORATION (US) 1984-07-31 US claimed
EP-1945705-A1 PHOTOLATENT SYSTEMS Ciba Holding Inc. (CH) 2008-07-23 EP disclosed
WO-2007054446-A1 PHOTOLATENT SYSTEMS CIBA HOLDING INC. (CH) 2007-05-18 WO disclosed
EP-0163635-A4 PROCESS FOR PREPARING SUBSTITUTED BENZYL MALONIC ACID ESTERS. ETHYL CORP (US) 1986-04-02 EP disclosed
EP-0163635-A1 PROCESS FOR PREPARING SUBSTITUTED BENZYL MALONIC ACID ESTERS ETHYL CORPORATION (US) 1985-12-11 EP disclosed
WO-1985002182-A1 PROCESS FOR PREPARING SUBSTITUTED BENZYL MALONIC ACID ESTERS ETHYL CORPORATION (US) 1985-05-23 WO disclosed
US-4463187-A Process for the preparation of 3,5-dihydrocarbyl-4-hydroxybenzylmalonic acid esters ETHYL CORPORATION (US) 1984-07-31 US disclosed