SCHEMBL4595237

SCHEMBL4595237

O=C1NCc2cc(-c3ccc(C(F)(F)F)cc3)ccc2N1.O=S1(=O)N=Cc2cc(-c3ccc(C(F)(F)F)cc3)ccc2N1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KIF11 P52732 3/20 0.47
CYP11B1 P15538 4/20 0.45
CYP11B2 P19099 4/20 0.45
TDP2 O95551 1/20 0.39
PDE3B Q13370 3/20 0.37
PDE3A Q14432 3/20 0.37
CA9 Q16790 3/20 0.36
GRIA1 P42261 1/20 0.35
CA12 O43570 2/20 0.34
AKT1 P31749 3/20 0.34
CDK2 P24941 2/20 0.34
CDK1 P06493 1/20 0.34
KIT P10721 1/20 0.34
KDR P35968 1/20 0.34
GRM2 Q14416 1/20 0.32
MAPK1 P28482 1/20 0.32
CYP1A2 P05177 2/20 0.32
CYP2C9 P11712 1/20 0.31
TBXAS1 P24557 1/20 0.31
MET P08581 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4896788 0.84 CA9 (0.45) KIF11TDP2CA9CA12
SCHEMBL4596154 0.83 KIF11 (0.41) KIF11TDP2CA9CA12AKT1
SCHEMBL4596437 0.83 KIF11 (0.65) KIF11CYP11B1CYP11B2TDP2PDE3B
SCHEMBL15966047 0.74 METAP2 (0.36) KIF11CA9CA12
SCHEMBL4889182 0.71 KIF11 (0.70) KIF11CYP11B1CYP11B2TDP2PDE3B
SCHEMBL4596526 0.69 KIF11 (0.57) KIF11CYP11B1CYP11B2TDP2PDE3B
SCHEMBL4596034 0.68 KIF11 (0.52) KIF11TDP2CA9CA12
SCHEMBL4898372 0.68 KIF11 (0.72) KIF11CYP11B1CYP11B2TDP2PDE3B
SCHEMBL1903306 0.67 KIF11 (0.80) KIF11CYP11B1CYP11B2TDP2PDE3B
SCHEMBL4897633 0.66 KIF11 (0.57) KIF11TDP2PDE3BPDE3ACA9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1874753-A2 COMPOUNDS, COMPOSITIONS AND METHODS SMITHKLINE BEECHAM CORPORATION (US) 2008-01-09 EP claimed
WO-2006113432-A2 COMPOUNDS, COMPOSITIONS AND METHODS SMITHKLINE BEECHAM CORPORATION (US) 2006-10-26 WO claimed