SCHEMBL4596154

SCHEMBL4596154

O=S1(=O)N=Cc2cc(-c3ccc(C(F)(F)F)cc3)ccc2N1.O=S1(=O)NCc2cc(-c3ccc(C(F)(F)F)cc3)ccc2N1

nearest known ligand 0.41

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
KIF11 P52732 1/20 0.41
CA9 Q16790 3/20 0.38
CA12 O43570 2/20 0.36
TDP2 O95551 1/20 0.36
AKT1 P31749 3/20 0.32
CDK2 P24941 2/20 0.32
CDK1 P06493 1/20 0.32
KIT P10721 1/20 0.32
KDR P35968 1/20 0.32
CHRNB2 P17787 1/20 0.31
CHRNA4 P43681 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4896788 0.86 CA9 (0.45) KIF11CA9CA12TDP2
SCHEMBL4596034 0.86 KIF11 (0.52) KIF11CA9CA12TDP2CHRNB2
SCHEMBL4595237 0.83 KIF11 (0.47) KIF11CA9CA12TDP2AKT1
SCHEMBL15966047 0.76 METAP2 (0.36) KIF11CA9CA12
SCHEMBL4898485 0.67 KIF11 (0.59) KIF11CA9CA12TDP2AKT1
SCHEMBL6911317 0.66 CYP11B2 (0.42)
SCHEMBL6910702 0.65 CYP11B1 (0.60) TDP2
SCHEMBL4596437 0.62 KIF11 (0.65) KIF11TDP2AKT1CDK2CDK1
SCHEMBL4897633 0.62 KIF11 (0.57) KIF11CA9CA12TDP2AKT1
SCHEMBL28061563 0.62 KIF11 (0.46) KIF11CA9CA12TDP2CHRNB2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1874753-A2 COMPOUNDS, COMPOSITIONS AND METHODS SMITHKLINE BEECHAM CORPORATION (US) 2008-01-09 EP disclosed
WO-2006113432-A2 COMPOUNDS, COMPOSITIONS AND METHODS SMITHKLINE BEECHAM CORPORATION (US) 2006-10-26 WO disclosed