SCHEMBL4595340

SCHEMBL4595340

Cc1cc2c(c(-c3cc(Cl)ccc3Cl)c1)OC(CN(CCc1ccccc1)C(=O)O)C2

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SIRT2 Q8IXJ6 1/20 0.36
AQP1 P29972 2/20 0.36
S1PR4 O95977 3/20 0.35
KDM4E B2RXH2 3/20 0.34
MAPK1 P28482 2/20 0.34
LPAR1 Q92633 2/20 0.34
ALDH1A1 P00352 2/20 0.34
RECQL P46063 1/20 0.34
LPAR2 Q9HBW0 1/20 0.34
MAPT P10636 4/20 0.34
MEN1 O00255 2/20 0.34
KMT2A Q03164 2/20 0.34
ATM Q13315 1/20 0.34
LPAR5 Q9H1C0 1/20 0.34
HTT P42858 2/20 0.33
OPRM1 P35372 1/20 0.33
OPRD1 P41143 1/20 0.33
TP53 P04637 1/20 0.33
L3MBTL1 Q9Y468 1/20 0.33
SMN1; SMN2 Q16637 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4596610 0.93 SIRT2 (0.40) SIRT2AQP1LPAR1ALDH1A1MAPT
SCHEMBL6367685 0.84 AQP1 (0.46) AQP1MAPTMEN1KMT2ATP53
SCHEMBL4231582 0.83 AQP1 (0.40) AQP1S1PR4KDM4EALDH1A1MAPT
SCHEMBL4595335 0.82 GPBAR1 (0.36) AQP1S1PR4ALDH1A1MAPTMEN1
SCHEMBL4596631 0.82 AQP1 (0.57) SIRT2AQP1KDM4ELPAR1ALDH1A1
SCHEMBL4596313 0.81 S1PR2 (0.38) AQP1S1PR4LPAR1ALDH1A1LPAR2
SCHEMBL4225416 0.79 MEN1 (0.37) SIRT2AQP1MEN1KMT2ATMEM97
SCHEMBL4831109 0.79 AQP1 (0.40) SIRT2AQP1S1PR4KDM4E
SCHEMBL4596351 0.79 AQP1 (0.45) AQP1KDM4EMAPK1MAPTMEN1
SCHEMBL4596674 0.79 SIRT2 (0.39) SIRT2AQP1LPAR1MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1874750-A1 DIHYDROBENZOFURANYL ALKANAMINE DERIVATIVES AS 5HT2C AGONISTS Wyeth Incoporated (US) 2008-01-09 EP disclosed