SCHEMBL4596610

SCHEMBL4596610

O=C(O)N(CCc1ccccc1)CC1Cc2cc(Cl)cc(-c3cc(Cl)ccc3Cl)c2O1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SIRT2 Q8IXJ6 1/20 0.40
AQP1 P29972 2/20 0.37
LPAR1 Q92633 2/20 0.36
LPAR5 Q9H1C0 2/20 0.36
MEN1 O00255 3/20 0.35
KMT2A Q03164 3/20 0.35
ALDH1A1 P00352 1/20 0.35
MAPT P10636 1/20 0.35
HTT P42858 1/20 0.35
SMN1; SMN2 Q16637 1/20 0.35
NPSR1 Q6W5P4 1/20 0.35
NPC1 O15118 1/20 0.34
RAB9A P51151 1/20 0.34
TDP1 Q9NUW8 1/20 0.34
GRIN2B Q13224 1/20 0.34
OPRM1 P35372 1/20 0.33
OPRD1 P41143 1/20 0.33
SCN5A Q14524 1/20 0.33
SCN2A Q99250 1/20 0.33
C5AR1 P21730 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4595340 0.93 SIRT2 (0.36) SIRT2AQP1LPAR1LPAR5MEN1
SCHEMBL4596631 0.85 AQP1 (0.57) SIRT2AQP1LPAR1LPAR5MEN1
SCHEMBL6368238 0.84 AQP1 (0.47) SIRT2AQP1MEN1KMT2AALDH1A1
SCHEMBL4596674 0.83 SIRT2 (0.39) SIRT2AQP1LPAR1LPAR5MEN1
SCHEMBL4225416 0.82 MEN1 (0.37) SIRT2AQP1MEN1KMT2ATMEM97
SCHEMBL4596313 0.82 S1PR2 (0.38) AQP1LPAR1MEN1KMT2AALDH1A1
SCHEMBL4220872 0.81 AQP1 (0.42) SIRT2AQP1MEN1KMT2ACNR2
SCHEMBL4596601 0.80 MEN1 (0.36) SIRT2AQP1MEN1KMT2AALDH1A1
SCHEMBL4229920 0.80 AQP1 (0.45) SIRT2AQP1LPAR1LPAR5MEN1
SCHEMBL5002222 0.80 OXTR (0.42) SIRT2MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1874750-A1 DIHYDROBENZOFURANYL ALKANAMINE DERIVATIVES AS 5HT2C AGONISTS Wyeth Incoporated (US) 2008-01-09 EP disclosed