SCHEMBL4596679

SCHEMBL4596679

Clc1cccc(Cl)c1-c1cccc2c1OC(CCc1ccccc1)C2

nearest known ligand 0.50

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
SIRT2 Q8IXJ6 2/20 0.50
AQP1 P29972 1/20 0.45
CYP3A4 P08684 2/20 0.40
SLC6A2 P23975 1/20 0.37
SLC6A4 P31645 1/20 0.37
SLC6A3 Q01959 1/20 0.37
PRKAB2 O43741 2/20 0.36
PRKAG1 P54619 2/20 0.36
PRKAA2 P54646 2/20 0.36
PRKAA1 Q13131 2/20 0.36
PRKAG3 Q9UGI9 2/20 0.36
PRKAG2 Q9UGJ0 2/20 0.36
PRKAB1 Q9Y478 2/20 0.36
DRD4 P21917 3/20 0.36
CYP1A2 P05177 1/20 0.35
CYP2D6 P10635 1/20 0.35
CYP2C9 P11712 1/20 0.35
SSTR2 P30874 1/20 0.34
SSTR4 P31391 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4595085 0.93 SIRT2 (0.54) SIRT2AQP1CYP3A4PRKAB2PRKAG1
SCHEMBL4596403 0.91 SIRT2 (0.48) SIRT2AQP1CYP3A4SLC6A2SLC6A4
SCHEMBL6047946 0.89 SIRT2 (0.46) SIRT2AQP1CYP3A4SLC6A2SLC6A4
SCHEMBL4595484 0.84 AQP1 (0.51) SIRT2AQP1CYP3A4SLC6A2SLC6A4
SCHEMBL4596728 0.83 SIRT2 (0.52) SIRT2AQP1CYP3A4PRKAB2PRKAG1
SCHEMBL4596777 0.83 SIRT2 (0.49) SIRT2AQP1CYP3A4PRKAB2PRKAG1
SCHEMBL4232135 0.83 AQP1 (0.47) SIRT2AQP1SLC6A2SLC6A4SLC6A3
SCHEMBL6047969 0.82 CYP3A4 (0.44) SIRT2CYP3A4SLC6A2SLC6A4SLC6A3
SCHEMBL12579303 0.80 PRKAB2 (0.54) AQP1PRKAB2PRKAG1PRKAA2PRKAA1
SCHEMBL4219827 0.80 PRKAB2 (0.54) AQP1PRKAB2PRKAG1PRKAA2PRKAA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1874750-A1 DIHYDROBENZOFURANYL ALKANAMINE DERIVATIVES AS 5HT2C AGONISTS Wyeth Incoporated (US) 2008-01-09 EP disclosed
EP-1675840-A1 DIHYDROBENZOFURANYL ALKANAMINE DERIVATIVES AS 5HT2C AGONISTS Wyeth a Corporation of the State of Delaware (US) 2006-07-05 EP disclosed
WO-2005044812-A1 DIHYDROBENZOFURANYL ALKANAMINE DERIVATIVES AS 5HT2C AGONISTS WYETH A CORPORATION OF THE STATE OF DELAWARE (US) 2005-05-19 WO disclosed