SCHEMBL4596289

SCHEMBL4596289

CC(C)(C)C(CC(O)c1ccccc1Cl)NC(=O)O

nearest known ligand 0.51

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
ADRB2 P07550 2/20 0.51
ADRB1 P08588 2/20 0.51
CYP2D6 P10635 1/20 0.51
NFKB1 P19838 1/20 0.51
HIF1A Q16665 1/20 0.51
BLM P54132 1/20 0.50
AOC3 Q16853 1/20 0.46
CASP1 P29466 1/20 0.40
CTSA P10619 4/20 0.39
CXCL8 P10145 2/20 0.38
MME P08473 1/20 0.36
ACE P12821 1/20 0.36
OPRM1 P35372 1/20 0.36
KMT2A Q03164 1/20 0.36
FDFT1 P37268 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4596259 0.83 CNR2 (0.43) ADRB2ADRB1HIF1ACTSAMME
SCHEMBL4595044 0.81 RIPK1 (0.45) AOC3MMEACE
SCHEMBL4596291 0.81 RIPK1 (0.45) AOC3MMEACE
SCHEMBL4389472 0.81 RIPK1 (0.45) AOC3MMEACE
SCHEMBL4595990 0.77 AOC3 (0.43) CYP2D6AOC3KMT2A
SCHEMBL4595463 0.76 ADRB3 (0.44) ADRB2ADRB1CYP2D6KMT2A
SCHEMBL4595555 0.75 POLB (0.39) CTSA
SCHEMBL1529699 0.72 NPC1 (0.45) BLMMMEACEKMT2A
SCHEMBL2532623 0.72 TDP1 (0.44) ADRB2NFKB1HIF1ABLMMME
SCHEMBL836126 0.72 ADRB2 (0.44) ADRB2ADRB1CYP2D6NFKB1HIF1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1874768-A2 INHIBITORS OF AKT ACTIVITY SMITHKLINE BEECHAM CORPORATION (US) 2008-01-09 EP disclosed
WO-2006113837-A2 INHIBITORS OF AKT ACTIVITY SMITHKLINE BEECHAM CORPORATION (US) 2006-10-26 WO disclosed