SCHEMBL4595463

SCHEMBL4595463

CC(C)(C)C(CC(O)c1cccc(Cl)c1)NC(=O)O

nearest known ligand 0.50

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
ADRB3 P13945 14/20 0.44
ADRB1 P08588 12/20 0.44
ADRB2 P07550 7/20 0.44
MEN1 O00255 1/20 0.42
KMT2A Q03164 1/20 0.42
ADRA1D P25100 1/20 0.41
ADRA1A P35348 1/20 0.41
ADRA1B P35368 1/20 0.41
CYP1A2 P05177 1/20 0.41
CYP2D6 P10635 1/20 0.41
CYP2C9 P11712 1/20 0.41
CYP2C19 P33261 1/20 0.41
KYNU Q16719 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4596291 0.84 RIPK1 (0.45)
SCHEMBL4595044 0.84 RIPK1 (0.45)
SCHEMBL4389472 0.84 RIPK1 (0.45)
SCHEMBL4595990 0.83 AOC3 (0.43) MEN1KMT2ACYP2D6CYP2C9CYP2C19
SCHEMBL4596066 0.82 L3MBTL1 (0.53) MEN1KMT2A
SCHEMBL2532623 0.76 TDP1 (0.44) ADRB2MEN1KMT2ACYP1A2CYP2C9
SCHEMBL4596289 0.76 ADRB2 (0.51) ADRB1ADRB2KMT2ACYP2D6
SCHEMBL23272194 0.73 MEN1 (0.43) ADRB3ADRB1MEN1KMT2ACYP2C19
SCHEMBL23272197 0.73 MEN1 (0.43) ADRB3ADRB1MEN1KMT2ACYP2C19
SCHEMBL4598598 0.73 S1PR3 (0.49) CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1874768-A2 INHIBITORS OF AKT ACTIVITY SMITHKLINE BEECHAM CORPORATION (US) 2008-01-09 EP disclosed
WO-2006113837-A2 INHIBITORS OF AKT ACTIVITY SMITHKLINE BEECHAM CORPORATION (US) 2006-10-26 WO disclosed