SCHEMBL4596574

SCHEMBL4596574

Cc1ccccc1-c1cccc2c1OC(N(C)C(=O)O)C2

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.40
MAPK1 P28482 1/20 0.40
SMN1; SMN2 Q16637 1/20 0.37
EDNRB P24530 1/20 0.35
EDNRA P25101 1/20 0.35
PARP1 P09874 3/20 0.35
SLC6A9 P48067 1/20 0.34
MYC P01106 1/20 0.33
KIF11 P52732 1/20 0.33
RAB9A P51151 2/20 0.33
MAPT P10636 2/20 0.33
NPC1 O15118 1/20 0.33
LMNA P02545 1/20 0.33
MCL1 Q07820 1/20 0.33
PRKAB2 O43741 1/20 0.32
PRKAG1 P54619 1/20 0.32
PRKAA2 P54646 1/20 0.32
PRKAA1 Q13131 1/20 0.32
PRKAG3 Q9UGI9 1/20 0.32
PRKAG2 Q9UGJ0 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4596236 0.90 MYC (0.39) ALDH1A1MAPK1SMN1; SMN2PARP1MYC
SCHEMBL4225937 0.87 HTR7 (0.43) ALDH1A1SMN1; SMN2PARP1PRKAB2PRKAG1
SCHEMBL4596973 0.86 HTR1A (0.41) ALDH1A1SMN1; SMN2PARP1SLC6A9KIF11
SCHEMBL4595391 0.86 HTR1A (0.41) ALDH1A1SMN1; SMN2PARP1SLC6A9KIF11
SCHEMBL4596752 0.85 RAB9A (0.38) ALDH1A1MAPK1SMN1; SMN2EDNRBEDNRA
SCHEMBL4597135 0.84 GPBAR1 (0.39) ALDH1A1MAPK1PARP1SLC6A9KIF11
SCHEMBL4236359 0.84 GPBAR1 (0.41) ALDH1A1MAPK1HTR2AHTR2C
SCHEMBL4230022 0.84 SMN1; SMN2 (0.35) SMN1; SMN2PARP1LMNA
SCHEMBL4596754 0.84 HTR7 (0.43) ALDH1A1EDNRBEDNRASLC6A9PRKAB2
SCHEMBL4226852 0.83 CNR2 (0.38) ALDH1A1SMN1; SMN2LMNAHTR2AHTR2C

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1874750-A1 DIHYDROBENZOFURANYL ALKANAMINE DERIVATIVES AS 5HT2C AGONISTS Wyeth Incoporated (US) 2008-01-09 EP disclosed
WO-2007030150-A1 DIHYDROBENZOFURANYL ALKANAMINE DERIVATIVES AS 5HT2C AGONISTS WYETH (US) 2007-03-15 WO disclosed
EP-1675840-A1 DIHYDROBENZOFURANYL ALKANAMINE DERIVATIVES AS 5HT2C AGONISTS Wyeth a Corporation of the State of Delaware (US) 2006-07-05 EP disclosed
WO-2005044812-A1 DIHYDROBENZOFURANYL ALKANAMINE DERIVATIVES AS 5HT2C AGONISTS WYETH A CORPORATION OF THE STATE OF DELAWARE (US) 2005-05-19 WO disclosed