SCHEMBL4596642

SCHEMBL4596642

COc1cc(Cl)cc2c1OC(C)C2

nearest known ligand 0.43

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.43
GAA P10253 2/20 0.43
SMN1; SMN2 Q16637 1/20 0.43
KLK7 P49862 1/20 0.41
KLK5 Q9Y337 1/20 0.41
KDM4E B2RXH2 4/20 0.39
PARP1 P09874 3/20 0.37
POLL Q9UGP5 1/20 0.37
HSD17B10 Q99714 2/20 0.37
HPGD P15428 1/20 0.37
ATM Q13315 1/20 0.37
EZH2 Q15910 1/20 0.35
MAP3K14 Q99558 1/20 0.34
HTR1A P08908 1/20 0.34
TSHR P16473 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4596639 0.82 EZH2 (0.35) ALDH1A1GAASMN1; SMN2ATMEZH2
SCHEMBL4597091 0.81 HTR2A (0.46) ALDH1A1GAASMN1; SMN2KDM4EPOLL
SCHEMBL15758805 0.80 ALDH1A1 (0.43) ALDH1A1GAASMN1; SMN2KLK7KLK5
SCHEMBL4597003 0.80 GPR84 (0.40) ALDH1A1GAASMN1; SMN2KLK7KLK5
SCHEMBL4220760 0.78 PRKAB2 (0.48) ATMEZH2MAP3K14
SCHEMBL4596514 0.78 CYP1A1 (0.41) ALDH1A1GAASMN1; SMN2KDM4EHSD17B10
SCHEMBL18768108 0.77 AKR1B1 (0.43) PARP1EZH2HTR1A
SCHEMBL4768067 0.77 KDM4E (0.39) ALDH1A1GAASMN1; SMN2KLK7KLK5
SCHEMBL14907125 0.75 TDP1 (0.52) ALDH1A1GAASMN1; SMN2KLK7KLK5
SCHEMBL12036045 0.74 PARP1 (0.48) GAAKLK7KLK5PARP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1874750-A1 DIHYDROBENZOFURANYL ALKANAMINE DERIVATIVES AS 5HT2C AGONISTS Wyeth Incoporated (US) 2008-01-09 EP disclosed
WO-2007030150-A1 DIHYDROBENZOFURANYL ALKANAMINE DERIVATIVES AS 5HT2C AGONISTS WYETH (US) 2007-03-15 WO disclosed