SCHEMBL4596652

SCHEMBL4596652

CN1Cc2cc(-c3ccc(C(F)(F)F)cc3)ccc2NC1=O.O=C1CSc2cc(-c3ccc4c(c3)OC(F)(F)O4)ccc2N1.OC1CCc2cc(-c3ccc(C(F)(F)F)cc3)ccc2C1

nearest known ligand 0.40

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
KIF11 P52732 3/20 0.40
TRPV1 Q8NER1 8/20 0.37
BRD4 O60885 2/20 0.35
BRD2 P25440 1/20 0.34
CREBBP Q92793 1/20 0.34
RORC P51449 1/20 0.34
PDE3B Q13370 2/20 0.33
PDE3A Q14432 2/20 0.33
TDP2 O95551 1/20 0.32
NTRK1 P04629 1/20 0.32
FLT3 P36888 1/20 0.32
NTRK3 Q16288 1/20 0.32
NTRK2 Q16620 1/20 0.32
CYP11B1 P15538 1/20 0.31
CYP11B2 P19099 1/20 0.31
MCHR1 Q99705 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4594863 0.97 KIF11 (0.39) KIF11TRPV1BRD4BRD2CREBBP
SCHEMBL4898840 0.72 CYP11B1 (0.53) KIF11PDE3BPDE3ACYP11B1CYP11B2
SCHEMBL4596440 0.71 KIF11 (0.63) KIF11TRPV1BRD4BRD2CREBBP
SCHEMBL4596362 0.70 KIF11 (0.61) KIF11PDE3BPDE3ATDP2CYP11B1
SCHEMBL4897709 0.69 CYP1A2 (0.55) KIF11TRPV1TDP2CYP11B1CYP11B2
SCHEMBL4596019 0.68 KIF11 (0.44) KIF11RORCPDE3BPDE3A
SCHEMBL4890586 0.66 KIF11 (0.58) KIF11PDE3BPDE3ACYP11B1CYP11B2
SCHEMBL4596493 0.64 NOTUM (0.47) KIF11PDE3BPDE3ACYP11B1CYP11B2
SCHEMBL27394981 0.63 BRD4 (0.62) KIF11TRPV1BRD4BRD2CREBBP
SCHEMBL22340014 0.63 BRD4 (0.56) KIF11BRD4BRD2CREBBPPDE3B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1874753-A2 COMPOUNDS, COMPOSITIONS AND METHODS SMITHKLINE BEECHAM CORPORATION (US) 2008-01-09 EP disclosed
WO-2006113432-A2 COMPOUNDS, COMPOSITIONS AND METHODS SMITHKLINE BEECHAM CORPORATION (US) 2006-10-26 WO disclosed