SCHEMBL4596728

SCHEMBL4596728

Clc1ccc(Cl)c(-c2cccc3c2OC(CCc2ccccc2)C3)c1

nearest known ligand 0.52

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
SIRT2 Q8IXJ6 2/20 0.52
AQP1 P29972 3/20 0.38
DRD4 P21917 2/20 0.37
CYP3A4 P08684 2/20 0.37
CYP1A2 P05177 1/20 0.37
CYP2D6 P10635 1/20 0.37
CYP2C9 P11712 1/20 0.37
SSTR2 P30874 1/20 0.36
SSTR4 P31391 1/20 0.36
PRKAB2 O43741 2/20 0.36
PRKAG1 P54619 2/20 0.36
PRKAA2 P54646 2/20 0.36
PRKAA1 Q13131 2/20 0.36
PRKAG3 Q9UGI9 2/20 0.36
PRKAG2 Q9UGJ0 2/20 0.36
PRKAB1 Q9Y478 2/20 0.36
CXCR2 P25025 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4596777 0.91 SIRT2 (0.49) SIRT2AQP1DRD4CYP3A4CYP1A2
SCHEMBL4596403 0.89 SIRT2 (0.48) SIRT2AQP1DRD4CYP3A4CYP1A2
SCHEMBL4595085 0.86 SIRT2 (0.54) SIRT2AQP1DRD4CYP3A4CYP1A2
SCHEMBL6047946 0.84 SIRT2 (0.46) SIRT2AQP1DRD4CYP3A4PRKAB2
SCHEMBL4596679 0.83 SIRT2 (0.50) SIRT2AQP1DRD4CYP3A4CYP1A2
SCHEMBL5795152 0.82 AQP1 (0.56) AQP1SSTR2SSTR4PRKAB2PRKAG1
SCHEMBL4226043 0.82 AQP1 (0.56) AQP1SSTR2SSTR4PRKAB2PRKAG1
SCHEMBL4596987 0.81 SIRT2 (0.55) SIRT2AQP1DRD4CYP3A4CYP1A2
SCHEMBL5148358 0.81 NFKB1 (0.43) SIRT2AQP1PRKAB2PRKAG1PRKAA2
SCHEMBL6047969 0.80 CYP3A4 (0.44) SIRT2DRD4CYP3A4PRKAB2PRKAG1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1874750-A1 DIHYDROBENZOFURANYL ALKANAMINE DERIVATIVES AS 5HT2C AGONISTS Wyeth Incoporated (US) 2008-01-09 EP disclosed