SCHEMBL4596693

SCHEMBL4596693

CC1Cc2cccc(C=Cc3ccccc3)c2O1

nearest known ligand 0.62

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
CREBBP Q92793 5/20 0.62
BRD4 O60885 4/20 0.62
PARP1 P09874 3/20 0.46
NFE2L2 Q16236 3/20 0.39
TRPA1 O75762 2/20 0.39
MAOA P21397 2/20 0.38
MAOB P27338 2/20 0.38
HTR1A P08908 3/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4596690 0.82 BRD4 (0.49) CREBBPBRD4NFE2L2TRPA1MAOA
SCHEMBL4228692 0.78 BRD4 (0.43) CREBBPBRD4NFE2L2TRPA1MAOA
SCHEMBL4228696 0.78 BRD4 (0.43) CREBBPBRD4NFE2L2TRPA1MAOA
SCHEMBL4230107 0.78 PARP1 (0.54) CREBBPBRD4PARP1MAOAMAOB
SCHEMBL17680709 0.77 CREBBP (1.00) CREBBPBRD4
SCHEMBL6047933 0.70 NFE2L2 (0.42) CREBBPBRD4NFE2L2TRPA1MAOA
SCHEMBL19122972 0.70 PARP1 (0.56) CREBBPBRD4PARP1MAOAMAOB
SCHEMBL13074639 0.70 PARP1 (0.56) CREBBPBRD4PARP1MAOAMAOB
SCHEMBL4596765 0.69 ALDH1A1 (0.48) CREBBPBRD4PARP1MAOAMAOB
SCHEMBL6047931 0.69 NFE2L2 (0.41) CREBBPBRD4NFE2L2TRPA1MAOA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1874750-A1 DIHYDROBENZOFURANYL ALKANAMINE DERIVATIVES AS 5HT2C AGONISTS Wyeth Incoporated (US) 2008-01-09 EP disclosed