SCHEMBL4596717

SCHEMBL4596717

O=C(CCOc1cc(-c2ccc(C(F)(F)F)cc2)ccc1[N+](=O)[O-])OCCCOc1cc(-c2ccc(C(F)(F)F)cc2)ccc1[N+](=O)[O-]

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP11B1 P15538 2/20 0.45
CYP11B2 P19099 2/20 0.45
GSTP1 P09211 1/20 0.42
GSTM2 P28161 1/20 0.42
ALDH1A1 P00352 5/20 0.39
TDP1 Q9NUW8 2/20 0.39
POLB P06746 1/20 0.38
PPARD Q03181 1/20 0.38
MAPT P10636 3/20 0.38
SMN1; SMN2 Q16637 2/20 0.38
NPC1 O15118 1/20 0.38
RAB9A P51151 1/20 0.38
LMNA P02545 1/20 0.37
CYP1A2 P05177 1/20 0.37
CYP3A4 P08684 1/20 0.37
CYP2D6 P10635 1/20 0.37
CYP2C9 P11712 1/20 0.37
CYP2C19 P33261 1/20 0.37
TTR P02766 2/20 0.37
HPGD P15428 2/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4596411 0.86 CYP11B1 (0.51) CYP11B1CYP11B2ALDH1A1TDP1POLB
SCHEMBL4890673 0.84 CYP11B1 (0.50) CYP11B1CYP11B2ALDH1A1POLBMAPT
SCHEMBL4596709 0.84 CYP11B1 (0.47) CYP11B1CYP11B2ALDH1A1TDP1POLB
SCHEMBL3903976 0.73 KIF11 (0.51) ALDH1A1TDP1MAPTSMN1; SMN2LMNA
SCHEMBL8354960 0.72 KMT2A (0.58) ALDH1A1TDP1POLBPPARDMAPT
SCHEMBL4898796 0.70 TTR (0.43) CYP11B1CYP11B2ALDH1A1TDP1POLB
SCHEMBL4596243 0.70 GSTP1 (0.53) GSTP1GSTM2ALDH1A1POLBMAPT
SCHEMBL4594932 0.70 MAPT (0.50) ALDH1A1POLBMAPTSMN1; SMN2NPC1
SCHEMBL4596633 0.69 MGLL (0.41) ALDH1A1TDP1POLBPPARDMAPT
SCHEMBL4594989 0.69 TTR (0.52) ALDH1A1TDP1MAPTCYP3A4TTR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1874753-A2 COMPOUNDS, COMPOSITIONS AND METHODS SMITHKLINE BEECHAM CORPORATION (US) 2008-01-09 EP disclosed
WO-2006113432-A2 COMPOUNDS, COMPOSITIONS AND METHODS SMITHKLINE BEECHAM CORPORATION (US) 2006-10-26 WO disclosed