SCHEMBL4596709

SCHEMBL4596709

O=C(O)CCOc1cc(-c2ccc(C(F)(F)F)cc2)ccc1[N+](=O)[O-].O=[N+]([O-])c1ccc(-c2ccc(C(F)(F)F)cc2)cc1OCCCO

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP11B1 P15538 2/20 0.47
CYP11B2 P19099 2/20 0.47
LTB4R Q15722 2/20 0.41
CHEK1 O14757 2/20 0.41
PTPN2 P17706 2/20 0.39
PTPN1 P18031 2/20 0.39
PTPN6 P29350 2/20 0.39
MEN1 O00255 1/20 0.38
TTR P02766 1/20 0.38
PPOX P50336 1/20 0.38
KMT2A Q03164 1/20 0.38
TDP1 Q9NUW8 1/20 0.38
POLB P06746 1/20 0.38
KDM4E B2RXH2 1/20 0.37
ALDH1A1 P00352 1/20 0.37
PPARD Q03181 2/20 0.37
PTGDR2 Q9Y5Y4 2/20 0.37
PPARA Q07869 1/20 0.37
ALOX5 P09917 1/20 0.37
PSEN1 P49768 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4596411 0.94 CYP11B1 (0.51) CYP11B1CYP11B2LTB4RPTPN2PTPN1
SCHEMBL4890673 0.92 CYP11B1 (0.50) CYP11B1CYP11B2CHEK1POLBALDH1A1
SCHEMBL4596717 0.84 CYP11B1 (0.45) CYP11B1CYP11B2CHEK1MEN1TTR
SCHEMBL4595112 0.76 HDAC2 (0.47) LTB4RPTPN2PTPN1PTPN6MEN1
SCHEMBL3903976 0.72 KIF11 (0.51) CHEK1MEN1KMT2ATDP1ALDH1A1
SCHEMBL4898796 0.72 TTR (0.43) CYP11B1CYP11B2CHEK1MEN1TTR
SCHEMBL29182839 0.71 NPC1 (0.44) CYP11B1CYP11B2MEN1KMT2APOLB
SCHEMBL19175209 0.71 MASP2 (0.51) MEN1KMT2ATDP1ALDH1A1PPARD
SCHEMBL30930995 0.71 NPC1 (0.44) CYP11B1CYP11B2MEN1KMT2APOLB
SCHEMBL3484477 0.71 ALDH1A1 (0.52) MEN1KMT2ATDP1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1874753-A2 COMPOUNDS, COMPOSITIONS AND METHODS SMITHKLINE BEECHAM CORPORATION (US) 2008-01-09 EP disclosed
WO-2006113432-A2 COMPOUNDS, COMPOSITIONS AND METHODS SMITHKLINE BEECHAM CORPORATION (US) 2006-10-26 WO disclosed