SCHEMBL4597055

SCHEMBL4597055

COc1cccc(-c2cccc3c2OC(C)C3)c1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR1A P08908 1/20 0.49
HTR7 P34969 1/20 0.49
PRKAB2 O43741 1/20 0.46
PRKAG1 P54619 1/20 0.46
PRKAA2 P54646 1/20 0.46
PRKAA1 Q13131 1/20 0.46
PRKAG3 Q9UGI9 1/20 0.46
PRKAG2 Q9UGJ0 1/20 0.46
PRKAB1 Q9Y478 1/20 0.46
LMNA P02545 2/20 0.46
GRM2 Q14416 1/20 0.44
CD274 Q9NZQ7 1/20 0.43
PARP1 P09874 3/20 0.43
CYP1A1 P04798 1/20 0.42
CYP1A2 P05177 1/20 0.42
CYP2E1 P05181 1/20 0.42
CYP3A4 P08684 1/20 0.42
CYP2C8 P10632 1/20 0.42
CYP2D6 P10635 1/20 0.42
CYP2A6 P11509 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4596788 0.87 DRD2 (0.52) HTR1AHTR7PRKAB2PRKAG1PRKAA2
SCHEMBL4597054 0.85 HTR1A (0.48) HTR1AHTR7PRKAB2PRKAG1PRKAA2
SCHEMBL4710706 0.84 PARP1 (0.43) HTR1AHTR7LMNAGRM2PARP1
SCHEMBL6047913 0.84 GPR84 (0.45) HTR1AHTR7LMNAGRM2CD274
SCHEMBL4220641 0.82 PRKAB2 (0.69) HTR1AHTR7PRKAB2PRKAG1PRKAA2
SCHEMBL4596822 0.81 KDM4E (0.44) HTR1AHTR7GRM2CYP1A1CYP1A2
SCHEMBL4713158 0.81 HDAC4 (0.43) PRKAB2PRKAG1PRKAA2PRKAA1PRKAG3
SCHEMBL4596518 0.81 CYP1A1 (0.50) PRKAB2PRKAG1PRKAA2PRKAA1PRKAG3
SCHEMBL4625851 0.80 HTR1A (0.47) HTR1AHTR7PRKAB2PRKAG1PRKAA2
SCHEMBL4624027 0.80 PRKAB2 (0.52) HTR1AHTR7PRKAB2PRKAG1PRKAA2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1874750-A1 DIHYDROBENZOFURANYL ALKANAMINE DERIVATIVES AS 5HT2C AGONISTS Wyeth Incoporated (US) 2008-01-09 EP disclosed
WO-2007030150-A1 DIHYDROBENZOFURANYL ALKANAMINE DERIVATIVES AS 5HT2C AGONISTS WYETH (US) 2007-03-15 WO disclosed
EP-1675840-A1 DIHYDROBENZOFURANYL ALKANAMINE DERIVATIVES AS 5HT2C AGONISTS Wyeth a Corporation of the State of Delaware (US) 2006-07-05 EP disclosed
WO-2005044812-A1 DIHYDROBENZOFURANYL ALKANAMINE DERIVATIVES AS 5HT2C AGONISTS WYETH A CORPORATION OF THE STATE OF DELAWARE (US) 2005-05-19 WO disclosed