SCHEMBL4597782

SCHEMBL4597782

O=C(O)N1CCC(NCC(NC2CCOCC2)c2ccccc2)CC1

nearest known ligand 0.42

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 1/20 0.42
CYP2C19 P33261 1/20 0.42
KDM4E B2RXH2 1/20 0.41
ALDH1A1 P00352 3/20 0.40
MEN1 O00255 1/20 0.38
KMT2A Q03164 1/20 0.38
AURKA O14965 1/20 0.37
RPS6KB1 P23443 1/20 0.37
DRD2 P14416 1/20 0.37
DRD4 P21917 1/20 0.37
DRD3 P35462 1/20 0.37
SMN1; SMN2 Q16637 1/20 0.37
TSHR P16473 1/20 0.36
PRMT5 O14744 2/20 0.36
HPGD P15428 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4023399 0.88 CCR5 (0.43)
SCHEMBL5575420 0.85 GPR119 (0.48) KDM4EALDH1A1SMN1; SMN2
SCHEMBL3754554 0.85 GPR119 (0.48) KDM4EALDH1A1SMN1; SMN2
SCHEMBL4206072 0.76 ATM (0.42) KDM4EALDH1A1TSHR
SCHEMBL18539369 0.75 KDM4E (0.43) KDM4EAURKARPS6KB1
SCHEMBL4609867 0.74 C3AR1 (0.42) CYP3A4CYP2C19KDM4EDRD3TSHR
SCHEMBL5576515 0.73 EPHX1 (0.53) KDM4EALDH1A1
SCHEMBL8311276 0.73 SOS1 (0.58) KDM4EMEN1KMT2ADRD2DRD4
SCHEMBL3763458 0.72 CTSK (0.44) KDM4EALDH1A1MEN1KMT2ASMN1; SMN2
SCHEMBL15520799 0.71 GAA (0.63)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1924265-A2 CHEMOKINE RECEPTOR BINDING COMPOUNDS Genzyme Corporation (US) 2008-05-28 EP disclosed
WO-2007022371-A2 CHEMOKINE RECEPTOR BINDING COMPOUNDS GENZYME CORPORATION (US) 2007-02-22 WO disclosed