SCHEMBL4597866

SCHEMBL4597866

Cc1ccc(F)c([C@@](I)(CO)NC(=O)OC(C)(C)C)c1

nearest known ligand 0.40

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
AAK1 Q2M2I8 12/20 0.40
KDR P35968 2/20 0.35
FLT1 P17948 1/20 0.35
AKT1 P31749 1/20 0.34
NPC1 O15118 1/20 0.34
MAPT P10636 1/20 0.34
RAB9A P51151 1/20 0.34
SMN1; SMN2 Q16637 1/20 0.34
TRPA1 O75762 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17118647 0.77 AAK1 (0.37) AAK1KDRFLT1MAPT
SCHEMBL17118650 0.77 AAK1 (0.38) AAK1KDRFLT1
SCHEMBL4597509 0.76 LMNA (0.40) AAK1AKT1MAPT
SCHEMBL3710918 0.74 CTSS (0.41) AAK1AKT1NPC1RAB9ASMN1; SMN2
SCHEMBL24944947 0.73 EPAS1 (0.39) AAK1
SCHEMBL4595970 0.72 CTSL (0.41) AKT1NPC1MAPTRAB9ASMN1; SMN2
SCHEMBL27945122 0.72 AAK1 (0.38) AAK1TRPA1
SCHEMBL253236 0.72 AAK1 (0.50) AAK1NPC1RAB9ASMN1; SMN2
SCHEMBL27945123 0.72 AAK1 (0.50) AAK1NPC1RAB9ASMN1; SMN2
SCHEMBL15315931 0.72 AAK1 (0.38) AAK1TRPA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1924265-A2 CHEMOKINE RECEPTOR BINDING COMPOUNDS Genzyme Corporation (US) 2008-05-28 EP disclosed
WO-2007022371-A2 CHEMOKINE RECEPTOR BINDING COMPOUNDS GENZYME CORPORATION (US) 2007-02-22 WO disclosed