SCHEMBL4598844

SCHEMBL4598844

CON1c2ccc(CP(=O)(O)O)cc2C(C)(C)C2COc3ccccc3C21

nearest known ligand 0.34

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
HCRTR1 O43613 2/20 0.34
HCRTR2 O43614 2/20 0.34
HSP90AA1 P07900 4/20 0.33
HTR2B P41595 1/20 0.32
ALDH1A1 P00352 1/20 0.32
GAA P10253 1/20 0.32
L3MBTL1 Q9Y468 1/20 0.32
MEN1 O00255 1/20 0.32
KMT2A Q03164 1/20 0.32
PSMB5 P28074 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4658821 0.86 HCRTR1 (0.32) HCRTR1HCRTR2HSP90AA1HTR2BALDH1A1
SCHEMBL4563416 0.81 LTB4R (0.36) HCRTR1HCRTR2HSP90AA1HTR2BALDH1A1
SCHEMBL4629499 0.80 HSP90AA1 (0.39) HSP90AA1ALDH1A1GAAL3MBTL1KMT2A
SCHEMBL4564085 0.80 HSP90AA1 (0.39) HSP90AA1ALDH1A1GAAL3MBTL1MEN1
SCHEMBL4564083 0.80 TSHR (0.42) HCRTR1HCRTR2HSP90AA1HTR2BALDH1A1
SCHEMBL4564518 0.80 LTB4R (0.38) HCRTR1HCRTR2
SCHEMBL4627927 0.80 ALDH1A1 (0.37) HSP90AA1HTR2BALDH1A1GAAL3MBTL1
SCHEMBL4556263 0.80 ALDH1A1 (0.37) HSP90AA1HTR2BALDH1A1GAAL3MBTL1
SCHEMBL4564158 0.79 HTR2B (0.36) HSP90AA1HTR2BALDH1A1GAAL3MBTL1
SCHEMBL4658817 0.79 NAMPT (0.32) HSP90AA1PSMB5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1907395-A1 ABCA1 ELEVATING COMPOUNDS CV THERAPEUTICS, INC. (US) 2008-04-09 EP disclosed
WO-2007002867-A1 ABCA1 ELEVATING COMPOUNDS CV THERAPEUTICS, INC. (US) 2007-01-04 WO disclosed