SCHEMBL4629499

SCHEMBL4629499

CON1c2ccc(Br)cc2C(C)(C)[C@H]2COc3ccccc3[C@H]21

nearest known ligand 0.39

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
HSP90AA1 P07900 4/20 0.39
ALDH1A1 P00352 2/20 0.33
HTR2A P28223 1/20 0.33
DRD2 P14416 1/20 0.33
DRD3 P35462 1/20 0.33
GAA P10253 1/20 0.33
L3MBTL1 Q9Y468 1/20 0.33
TP53 P04637 1/20 0.33
MAPT P10636 1/20 0.33
KMT2A Q03164 1/20 0.33
SMN1; SMN2 Q16637 1/20 0.33
LMNA P02545 1/20 0.31
HTT P42858 1/20 0.31
CYP3A4 P08684 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4564085 0.86 HSP90AA1 (0.39) HSP90AA1ALDH1A1DRD2DRD3GAA
SCHEMBL4627927 0.86 ALDH1A1 (0.37) HSP90AA1ALDH1A1GAAL3MBTL1MAPT
SCHEMBL4556263 0.86 ALDH1A1 (0.37) HSP90AA1ALDH1A1GAAL3MBTL1MAPT
SCHEMBL4564158 0.85 HTR2B (0.36) HSP90AA1ALDH1A1GAAL3MBTL1
SCHEMBL4564188 0.84 LTB4R (0.34) HSP90AA1ALDH1A1GAAL3MBTL1CYP3A4
SCHEMBL4564453 0.84 HSP90AA1 (0.34) HSP90AA1ALDH1A1HTR2AGAAL3MBTL1
SCHEMBL4627857 0.84 ALDH1A1 (0.32) HSP90AA1ALDH1A1GAAL3MBTL1CYP3A4
SCHEMBL4658821 0.84 HCRTR1 (0.32) HSP90AA1ALDH1A1HTR2ADRD2DRD3
SCHEMBL4564019 0.84 LMNA (0.38) HSP90AA1ALDH1A1GAAL3MBTL1MAPT
SCHEMBL4564341 0.83 HSD11B1 (0.39) DRD2DRD3MAPTKMT2ASMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1907395-A1 ABCA1 ELEVATING COMPOUNDS CV THERAPEUTICS, INC. (US) 2008-04-09 EP disclosed
WO-2007002867-A1 ABCA1 ELEVATING COMPOUNDS CV THERAPEUTICS, INC. (US) 2007-01-04 WO disclosed