SCHEMBL4564158

SCHEMBL4564158

CON1c2ccc(-c3ccccc3)cc2C(C)(C)[C@@H]2COc3ccccc3[C@H]21

nearest known ligand 0.36

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
HTR2B P41595 2/20 0.36
TMEM97 Q5BJF2 2/20 0.36
SIGMAR1 Q99720 2/20 0.36
HTR1A P08908 1/20 0.36
HTR7 P34969 1/20 0.35
HSP90AA1 P07900 1/20 0.34
CHRNB4 P30926 2/20 0.33
CHRNA3 P32297 2/20 0.33
L3MBTL1 Q9Y468 2/20 0.33
ALDH1A1 P00352 1/20 0.33
GAA P10253 1/20 0.33
BACE1 P56817 1/20 0.32
ADRA1D P25100 4/20 0.32
ADRA1A P35348 4/20 0.32
ADRA1B P35368 4/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4657250 0.93 LMNA (0.38) HSP90AA1L3MBTL1ALDH1A1GAABACE1
SCHEMBL4628825 0.91 RARB (0.39)
SCHEMBL4564228 0.90 CACNA1B (0.35)
SCHEMBL4564105 0.88 PDE4A (0.37) HTR2BHTR1A
SCHEMBL4563452 0.88 PTGS2 (0.39) L3MBTL1ALDH1A1GAAADRA1A
SCHEMBL4564518 0.87 LTB4R (0.38)
SCHEMBL4565660 0.86 PDK2 (0.41)
SCHEMBL4564085 0.85 HSP90AA1 (0.39) HSP90AA1L3MBTL1ALDH1A1GAA
SCHEMBL4629499 0.85 HSP90AA1 (0.39) HSP90AA1L3MBTL1ALDH1A1GAA
SCHEMBL4566254 0.85 PDK2 (0.41) L3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2125825-A1 ABCA1 ELEVATING COMPOUNDS CV THERAPEUTICS, INC. (US) 2009-12-02 EP disclosed
WO-2008079139-A1 ABCA1 ELEVATING COMPOUNDS CV THERAPEUTICS, INC. (US) 2008-07-03 WO disclosed