SCHEMBL4600433

SCHEMBL4600433

Cc1cc(CCn2c(C(=O)O)cc3cc(F)ccc32)ccn1

nearest known ligand 0.51

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.51
KDM4E B2RXH2 1/20 0.51
HPGD P15428 1/20 0.51
HSD17B10 Q99714 1/20 0.51
CCR2 P41597 6/20 0.49
IDO1 P14902 1/20 0.42
CYP1A2 P05177 1/20 0.40
POLB P06746 1/20 0.40
PLA2G4A P47712 3/20 0.40
MCL1 Q07820 3/20 0.39
NTRK1 P04629 2/20 0.37
GPR35 Q9HC97 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4599937 0.89 CCR2 (0.63) ALDH1A1KDM4EHPGDHSD17B10CCR2
SCHEMBL3615596 0.87 KDM4E (0.45) ALDH1A1KDM4EHPGDHSD17B10CCR2
SCHEMBL13802523 0.82 CCR2 (0.62) ALDH1A1KDM4EHPGDHSD17B10CCR2
SCHEMBL15362051 0.79 TP53 (0.35) ALDH1A1KDM4EHPGDHSD17B10IDO1
SCHEMBL4599686 0.79 IDO1 (0.61) ALDH1A1KDM4EHPGDHSD17B10CCR2
SCHEMBL4600294 0.77 ALDH1A1 (0.50) ALDH1A1KDM4EHPGDHSD17B10CCR2
SCHEMBL12466547 0.77 ALDH1A1 (0.66) ALDH1A1KDM4EHPGDHSD17B10CCR2
SCHEMBL3617356 0.76 MAPT (0.53) ALDH1A1KDM4EHPGDCCR2POLB
SCHEMBL4599709 0.76 CCR2 (0.55) ALDH1A1KDM4EHPGDHSD17B10CCR2
SCHEMBL2895007 0.75 CCR2 (0.70) ALDH1A1KDM4EHPGDHSD17B10CCR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1910335-A1 N-(HETEROARYL)-1-HETEROARYLALKYL-1H-INDOLE-2-CARBOXAMIDE DERIVATIVES, PREPARATION AND USE THEREOF Sanofi-Aventis (FR) 2008-04-16 EP claimed
WO-2007010144-A1 N-(HETEROARYL)-1-HETEROARYLALKYL-1H-INDOLE-2-CARBOXAMIDE DERIVATIVES, PREPARATION AND USE THEREOF SANOFI-AVENTIS (FR) 2007-01-25 WO claimed