SCHEMBL4600708

SCHEMBL4600708

CON(C)C(=O)[C@H](CNC(=O)O)c1ccccn1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP2C19 P33261 2/20 0.43
KCNA5 P22460 3/20 0.42
GAA P10253 2/20 0.40
MEN1 O00255 1/20 0.40
KMT2A Q03164 1/20 0.40
SMN1; SMN2 Q16637 1/20 0.40
TSHR P16473 3/20 0.39
ALDH1A1 P00352 3/20 0.39
LMNA P02545 2/20 0.39
CYP3A4 P08684 1/20 0.39
KDM4E B2RXH2 1/20 0.39
RAB9A P51151 1/20 0.39
CYP1A2 P05177 1/20 0.39
CHRM2 P08172 1/20 0.37
SLC6A2 P23975 1/20 0.37
SLC6A4 P31645 1/20 0.37
SCN1A P35498 1/20 0.37
SCN2A Q99250 1/20 0.37
SCN3A Q9NY46 1/20 0.37
PMP22 Q01453 2/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17825622 0.81 KMT2A (0.41) MEN1KMT2ATSHRALDH1A1LMNA
SCHEMBL4598534 0.76 MC4R (0.40) GAAMEN1KMT2AALDH1A1LMNA
SCHEMBL28583802 0.73 CYP2C19 (0.47) CYP2C19KCNA5GAAMEN1KMT2A
SCHEMBL23354438 0.72 ALDH1A1 (0.45) GAAMEN1KMT2ASMN1; SMN2ALDH1A1
SCHEMBL26906885 0.72 ALDH1A1 (0.45) GAAMEN1KMT2ASMN1; SMN2ALDH1A1
SCHEMBL6466556 0.71 MTNR1A (0.44) MEN1KMT2ANPSR1
SCHEMBL6342824 0.70 KCNA3 (0.42) KCNA5MEN1KMT2ASMN1; SMN2TSHR
SCHEMBL4600703 0.70 HDAC6 (0.48) KMT2ASMN1; SMN2TSHRLMNACYP3A4
SCHEMBL14737238 0.69 MMP9 (0.42) CYP2C19MEN1KMT2AALDH1A1CYP1A2
SCHEMBL30771400 0.68 MEN1 (0.46) CYP2C19GAAMEN1KMT2AALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1912946-A1 PYRIDINE DERIVATIVES AS DIPEPTEDYL PEPTIDASE INHIBITORS Eli Lilly and Company (US) 2008-04-23 EP disclosed
WO-2007015767-A1 PYRIDINE DERIVATIVES AS DIPEPTEDYL PEPTIDASE INHIBITORS ELI LILLY AND COMPANY (US) 2007-02-08 WO disclosed