SCHEMBL4598534

SCHEMBL4598534

CON(C)C(=O)[C@H](CNC(=O)O)c1ccccc1F

nearest known ligand 0.40

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
MC4R P32245 3/20 0.40
OPRM1 P35372 1/20 0.40
C5AR1 P21730 3/20 0.38
ALDH1A1 P00352 1/20 0.38
LMNA P02545 1/20 0.38
CNR2 P34972 1/20 0.37
MEN1 O00255 1/20 0.37
KMT2A Q03164 1/20 0.37
CTSA P10619 6/20 0.36
CES2 O00748 1/20 0.35
CES1 P23141 1/20 0.35
GAA P10253 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4597242 0.84 JAK3 (0.42) MC4ROPRM1ALDH1A1LMNA
SCHEMBL17825622 0.82 KMT2A (0.41) ALDH1A1LMNAMEN1KMT2A
SCHEMBL4600708 0.76 CYP2C19 (0.43) ALDH1A1LMNAMEN1KMT2AGAA
SCHEMBL4600313 0.75 KCNA5 (0.41) LMNAMEN1KMT2A
SCHEMBL4598809 0.74 CTSK (0.40) LMNAMEN1KMT2A
SCHEMBL4600484 0.74 CTSK (0.40) LMNAMEN1KMT2A
SCHEMBL6466556 0.72 MTNR1A (0.44) CNR2MEN1KMT2A
SCHEMBL26907022 0.71 PRMT3 (0.48) MC4ROPRM1LMNACNR2CES2
SCHEMBL6342824 0.71 KCNA3 (0.42) ALDH1A1MEN1KMT2A
SCHEMBL27881358 0.71 CES2 (0.37) MC4RALDH1A1LMNACNR2MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1912946-A1 PYRIDINE DERIVATIVES AS DIPEPTEDYL PEPTIDASE INHIBITORS Eli Lilly and Company (US) 2008-04-23 EP disclosed
WO-2007015767-A1 PYRIDINE DERIVATIVES AS DIPEPTEDYL PEPTIDASE INHIBITORS ELI LILLY AND COMPANY (US) 2007-02-08 WO disclosed