SCHEMBL4600968

SCHEMBL4600968

CC(C)(C)NC(=O)c1cccnc1C(Cc1cc(C(F)(F)F)ccc1F)C(=O)CNC(=O)OC(C)(C)C

nearest known ligand 0.37

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
ALOX5AP P20292 2/20 0.37
FEN1 P39748 2/20 0.37
ANO1 Q5XXA6 5/20 0.35
AURKB Q96GD4 1/20 0.35
RXFP1 Q9HBX9 1/20 0.35
SCN9A Q15858 1/20 0.34
SMN1; SMN2 Q16637 1/20 0.34
KDM4E B2RXH2 2/20 0.33
MEN1 O00255 1/20 0.33
CYP1A2 P05177 1/20 0.33
CYP2C19 P33261 1/20 0.33
KMT2A Q03164 1/20 0.33
NPSR1 Q6W5P4 1/20 0.33
FNTA P49354 2/20 0.33
FNTB P49356 2/20 0.33
RIPK1 Q13546 2/20 0.32
HPGD P15428 1/20 0.32
TRPM8 Q7Z2W7 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4600646 0.91 SCN9A (0.41) ALOX5APFEN1ANO1SCN9ASMN1; SMN2
SCHEMBL4632372 0.90 SCN9A (0.35) ALOX5APFEN1ANO1SCN9ASMN1; SMN2
SCHEMBL4602360 0.90 ANO1 (0.41) ANO1AURKBSCN9ASMN1; SMN2FNTA
SCHEMBL4601576 0.88 CTSS (0.42) ALOX5APFEN1ANO1SCN9ASMN1; SMN2
SCHEMBL4632696 0.80 CTSS (0.44) SCN9ASMN1; SMN2MEN1KMT2A
SCHEMBL267770 0.79 SCN9A (0.40) ALOX5APFEN1ANO1SCN9A
SCHEMBL268189 0.77 ALOX5AP (0.37) ALOX5APFEN1ANO1RXFP1SCN9A
SCHEMBL4602131 0.77 KCNA5 (0.40) SMN1; SMN2
SCHEMBL4837234 0.76 ANO1 (0.39) ANO1SMN1; SMN2
SCHEMBL4600309 0.75 SCN9A (0.43) ANO1AURKBSCN9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1912946-A1 PYRIDINE DERIVATIVES AS DIPEPTEDYL PEPTIDASE INHIBITORS Eli Lilly and Company (US) 2008-04-23 EP disclosed
WO-2007015767-A1 PYRIDINE DERIVATIVES AS DIPEPTEDYL PEPTIDASE INHIBITORS ELI LILLY AND COMPANY (US) 2007-02-08 WO disclosed