SCHEMBL4600646

SCHEMBL4600646

CC(C)(C)NC(=O)c1cccnc1C(Cc1cc(F)ccc1F)C(=O)CNC(=O)OC(C)(C)C

nearest known ligand 0.41

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
SCN9A Q15858 4/20 0.41
SCN10A Q9Y5Y9 2/20 0.35
CYP3A4 P08684 1/20 0.35
ALOX5AP P20292 2/20 0.35
FEN1 P39748 2/20 0.35
ANO1 Q5XXA6 5/20 0.34
SMN1; SMN2 Q16637 1/20 0.34
LMNA P02545 1/20 0.33
SGMS2 Q8NHU3 1/20 0.33
CTSS P25774 1/20 0.33
CTSK P43235 1/20 0.33
GPR119 Q8TDV5 1/20 0.33
ADRA1D P25100 1/20 0.33
ADRA1A P35348 1/20 0.33
ADRA1B P35368 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4602360 0.92 ANO1 (0.41) SCN9AANO1SMN1; SMN2
SCHEMBL4632372 0.92 SCN9A (0.35) SCN9ASCN10AALOX5APFEN1ANO1
SCHEMBL4600968 0.91 ALOX5AP (0.37) SCN9AALOX5APFEN1ANO1SMN1; SMN2
SCHEMBL4601576 0.91 CTSS (0.42) SCN9ASCN10ACYP3A4ALOX5APFEN1
SCHEMBL4600309 0.84 SCN9A (0.43) SCN9ASCN10ACYP3A4ANO1CTSS
SCHEMBL4632696 0.82 CTSS (0.44) SCN9ASCN10ACYP3A4SMN1; SMN2LMNA
SCHEMBL4597310 0.81 ANO1 (0.39) SCN9AANO1GPR119
SCHEMBL4602131 0.79 KCNA5 (0.40) SMN1; SMN2LMNA
SCHEMBL4598878 0.79 CTSS (0.43) SCN9ASCN10AALOX5APFEN1ANO1
SCHEMBL269249 0.78 SCN9A (0.48) SCN9ASCN10ACYP3A4ANO1CTSS

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1912946-A1 PYRIDINE DERIVATIVES AS DIPEPTEDYL PEPTIDASE INHIBITORS Eli Lilly and Company (US) 2008-04-23 EP disclosed
WO-2007015767-A1 PYRIDINE DERIVATIVES AS DIPEPTEDYL PEPTIDASE INHIBITORS ELI LILLY AND COMPANY (US) 2007-02-08 WO disclosed