SCHEMBL4601576

SCHEMBL4601576

CC(C)(C)NC(=O)c1cccnc1[C@@H](Cc1ccccc1F)C(=O)CNC(=O)OC(C)(C)C

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CTSS P25774 1/20 0.42
CTSK P43235 1/20 0.42
LMNA P02545 1/20 0.41
SCN9A Q15858 6/20 0.40
SCN10A Q9Y5Y9 2/20 0.40
ANO1 Q5XXA6 1/20 0.38
SMN1; SMN2 Q16637 1/20 0.37
NPC1 O15118 2/20 0.37
MEN1 O00255 1/20 0.37
RAB9A P51151 1/20 0.37
KMT2A Q03164 1/20 0.37
KCNA5 P22460 1/20 0.36
PTPN1 P18031 1/20 0.36
MAPK8 P45983 1/20 0.36
CYP3A4 P08684 2/20 0.35
GLA P06280 1/20 0.35
TSHR P16473 1/20 0.35
L3MBTL1 Q9Y468 1/20 0.35
ALOX5AP P20292 1/20 0.34
FEN1 P39748 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4632696 0.91 CTSS (0.44) CTSSCTSKLMNASCN9ASCN10A
SCHEMBL4600646 0.91 SCN9A (0.41) CTSSCTSKLMNASCN9ASCN10A
SCHEMBL4632372 0.90 SCN9A (0.35) CTSSCTSKLMNASCN9ASCN10A
SCHEMBL4602360 0.90 ANO1 (0.41) SCN9AANO1SMN1; SMN2
SCHEMBL4600968 0.88 ALOX5AP (0.37) SCN9AANO1SMN1; SMN2MEN1KMT2A
SCHEMBL4598878 0.81 CTSS (0.43) CTSSCTSKSCN9ASCN10AANO1
SCHEMBL4600120 0.81 CTSS (0.48) CTSSCTSKLMNASCN9ASCN10A
SCHEMBL4598164 0.80 CTSS (0.42) CTSSCTSKSCN9AANO1NPC1
SCHEMBL4602131 0.80 KCNA5 (0.40) LMNASMN1; SMN2RAB9AKCNA5TSHR
SCHEMBL4598249 0.80 CTSS (0.42) CTSSCTSKLMNASCN9AANO1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1912946-A1 PYRIDINE DERIVATIVES AS DIPEPTEDYL PEPTIDASE INHIBITORS Eli Lilly and Company (US) 2008-04-23 EP disclosed
WO-2007015767-A1 PYRIDINE DERIVATIVES AS DIPEPTEDYL PEPTIDASE INHIBITORS ELI LILLY AND COMPANY (US) 2007-02-08 WO disclosed