SCHEMBL4601022

SCHEMBL4601022

COC(=O)c1ccc(NC(=O)c2ccc3c(c2)NCCC3)cc1

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 7/20 0.51
RAB9A P51151 7/20 0.51
SMN1; SMN2 Q16637 4/20 0.51
CASP3 P42574 1/20 0.51
SENP7 Q9BQF6 1/20 0.51
PLAU P00749 1/20 0.51
KMT2A Q03164 4/20 0.50
ALDH1A1 P00352 3/20 0.50
MEN1 O00255 3/20 0.50
TP53 P04637 2/20 0.50
PKM P14618 2/20 0.50
HPGD P15428 1/20 0.50
MAPK1 P28482 1/20 0.50
L3MBTL1 Q9Y468 1/20 0.49
ATM Q13315 1/20 0.49
PTPN1 P18031 1/20 0.47
PIR O00625 1/20 0.47
GSK3B P49841 1/20 0.47
HSF1 Q00613 1/20 0.47
CTDSP1 Q9GZU7 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3566272 0.89 MAPT (0.56) NPC1RAB9ASMN1; SMN2PLAUKMT2A
SCHEMBL554225 0.87 MAPT (0.51) KMT2AALDH1A1MEN1HPGDMAPK1
SCHEMBL30955089 0.87 MAPT (0.51) KMT2AALDH1A1MEN1HPGDMAPK1
SCHEMBL3571433 0.86 PYGL (0.55) NPC1RAB9ASMN1; SMN2PLAUKMT2A
SCHEMBL3571275 0.81 RAB9A (0.57) NPC1RAB9ASMN1; SMN2KMT2AALDH1A1
SCHEMBL29906783 0.79 ALDH1A1 (0.47) SMN1; SMN2KMT2AALDH1A1MEN1TP53
SCHEMBL2898350 0.79 ALDH1A1 (0.47) SMN1; SMN2KMT2AALDH1A1MEN1TP53
SCHEMBL3574814 0.78 PYGL (0.47) NPC1RAB9ASMN1; SMN2PLAUKMT2A
SCHEMBL3576854 0.78 PYGL (0.47) NPC1RAB9ASMN1; SMN2PLAUKMT2A
Hydrochloric Acid SCHEMBL29940234 0.77 ALDH1A1 (0.46) SMN1; SMN2KMT2AALDH1A1MEN1TP53

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1926711-A1 NOVEL HETEROBICYCLIC DERIVATIVES USEFUL AS INHIBITORS OF LIVER CARNITINE PALMITOYL TRANSFERASE F.HOFFMANN-LA ROCHE AG (CH) 2008-06-04 EP disclosed
WO-2007031429-A1 NOVEL HETEROBICYCLIC DERIVATIVES USEFUL AS INHIBITORS OF LIVER CARNITINE PALMITOYL TRANSFERASE F. HOFFMANN-LA ROCHE AG (CH) 2007-03-22 WO disclosed