SCHEMBL4601784

SCHEMBL4601784

Cn1ccnc1CN1CCC(NC(=O)OC(C)(C)C)CC1

nearest known ligand 0.50

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
KCNA3 P22001 1/20 0.50
AKT1 P31749 1/20 0.46
NSD2 O96028 1/20 0.46
DRD2 P14416 5/20 0.45
DRD3 P35462 1/20 0.45
CKS1B P61024 1/20 0.44
SKP1 P63208 1/20 0.44
SKP2 Q13309 1/20 0.44
AAK1 Q2M2I8 2/20 0.43
CCR5 P51681 1/20 0.43
CTSK P43235 2/20 0.43
NAMPT P43490 1/20 0.42
KMT2A Q03164 1/20 0.42
L3MBTL1 Q9Y468 1/20 0.42
PARP1 P09874 1/20 0.41
PARP2 Q9UGN5 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL648348 0.79 SIGMAR1 (0.60) KCNA3AKT1NSD2DRD2KMT2A
SCHEMBL14223071 0.78 ALOX15 (0.49) KCNA3AKT1NSD2DRD2CKS1B
SCHEMBL1956790 0.78 CYP3A4 (0.49) KCNA3AKT1NSD2DRD2CKS1B
SCHEMBL7078816 0.78 DRD4 (0.58) KCNA3AKT1DRD2DRD3CKS1B
SCHEMBL2731871 0.78 GPR119 (0.45) NSD2CKS1BSKP1SKP2KMT2A
SCHEMBL26640819 0.77 KCNA3 (0.50) KCNA3AKT1NSD2DRD2DRD3
SCHEMBL1956090 0.76 KCNA3 (0.47) KCNA3AKT1NSD2DRD2DRD3
SCHEMBL915402 0.76 KMT2A (0.65) KCNA3DRD2DRD3KMT2AL3MBTL1
SCHEMBL24247901 0.75 KCNA3 (0.46) KCNA3AKT1NSD2DRD2CKS1B
SCHEMBL16854336 0.75 ALDH1A1 (0.55) KCNA3AKT1DRD2DRD3CKS1B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1914235-A1 CHIRAL TETRA-HYDRO BETA-CARBOLINE DERIVATIVES AND APPLICATIONS THEREOF AS ANTIPARASITIC COMPOUNDS Universite de Lille 2 Droit et Santé (FR) 2008-04-23 EP disclosed
EP-1914235-A1 CHIRAL TETRA-HYDRO BETA-CARBOLINE DERIVATIVES AND APPLICATIONS THEREOF AS ANTIPARASITIC COMPOUNDS Universite de Lille 2 Droit et Santé (FR) 2008-04-23 EP disclosed