SCHEMBL4601994

SCHEMBL4601994

CCCCOC(=O)NCC(CCC(=O)OCC(C)C)N(C)C

nearest known ligand 0.42

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
CHRNB2 P17787 3/20 0.42
CHRNB4 P30926 3/20 0.42
CHRNA3 P32297 3/20 0.42
CHRNA4 P43681 3/20 0.42
ACHE P22303 11/20 0.38
NPC1 O15118 2/20 0.38
RAB9A P51151 2/20 0.38
SMN1; SMN2 Q16637 2/20 0.38
LMNA P02545 2/20 0.38
HRH4 Q9H3N8 1/20 0.37
HRH3 Q9Y5N1 1/20 0.37
MAPT P10636 1/20 0.37
ALDH1A1 P00352 1/20 0.36
CYP3A4 P08684 1/20 0.36
TSHR P16473 1/20 0.36
ATM Q13315 1/20 0.36
TDP1 Q9NUW8 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4632009 0.87 CHRNB2 (0.43) CHRNB2CHRNB4CHRNA3CHRNA4ACHE
SCHEMBL4603603 0.80 CHRNB2 (0.38) CHRNB2CHRNB4CHRNA3CHRNA4ACHE
SCHEMBL28522595 0.73 ACHE (0.56) ACHENPC1RAB9ASMN1; SMN2LMNA
SCHEMBL11465997 0.72 MAPT (0.61) LMNAMAPTALDH1A1CYP3A4TSHR
SCHEMBL29024707 0.72 DGKA (0.51) LMNAMAPTALDH1A1
SCHEMBL29024902 0.72 DGKA (0.51) LMNAMAPTALDH1A1
SCHEMBL29024901 0.72 DGKA (0.51) LMNAMAPTALDH1A1
SCHEMBL29024897 0.72 DGKA (0.51) LMNAMAPTALDH1A1
SCHEMBL29024898 0.72 DGKA (0.51) LMNAMAPTALDH1A1
SCHEMBL1866206 0.71 MAPT (0.64) LMNAMAPTALDH1A1CYP3A4TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1915351-A1 QUINAZOLINE DERIVATIVES USEFUL IN CANCER TREATMENT SCHERING CORPORATION (US) 2008-04-30 EP disclosed
WO-2007011618-A1 QUINAZOLINE DERIVATIVES USEFUL IN CANCER TREATMENT SCHERING CORPORATION (US) 2007-01-25 WO disclosed