SCHEMBL4602522

SCHEMBL4602522

C#CCOC1CC(COc2ccccc2Cl)N(C(=O)OCCCC)C1

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
L3MBTL1 Q9Y468 3/20 0.36
TDP1 Q9NUW8 2/20 0.36
ALDH1A1 P00352 1/20 0.36
ITGB1 P05556 1/20 0.35
ITGA5 P08648 1/20 0.35
PPARG P37231 1/20 0.34
PPARD Q03181 1/20 0.34
PPARA Q07869 1/20 0.34
ECE1 P42892 1/20 0.34
PTGDR2 Q9Y5Y4 1/20 0.33
TSHR P16473 1/20 0.33
SSTR1 P30872 1/20 0.33
SSTR4 P31391 1/20 0.33
BCHE P06276 1/20 0.33
ITGA4 P13612 1/20 0.33
NPFFR1 Q9GZQ6 1/20 0.33
NPFFR2 Q9Y5X5 1/20 0.33
NPC1 O15118 2/20 0.33
RAB9A P51151 2/20 0.33
KMT2A Q03164 2/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2200981 0.84 ABCB1 (0.39) SSTR1SSTR4DPP4PREPFAP
SCHEMBL30580462 0.72 TSHR (0.48) L3MBTL1TDP1ALDH1A1ECE1TSHR
SCHEMBL29612789 0.68 LMNA (0.46) L3MBTL1TDP1ALDH1A1TSHRBCHE
SCHEMBL8703069 0.68 TP53 (0.40) PPARGECE1TSHRSMN1; SMN2ALOX15
SCHEMBL4602385 0.67 GPR119 (0.39) ALDH1A1TSHRSSTR1SSTR4KMT2A
SCHEMBL2202034 0.67 GPR119 (0.39) ALDH1A1TSHRSSTR1SSTR4KMT2A
SCHEMBL2199374 0.67 SLC6A4 (0.39) SSTR4DPP4PREPFAPDPP8
SCHEMBL2201807 0.66 POLB (0.42) TSHRSSTR1SSTR4KMT2ADPP4
SCHEMBL4603500 0.66 POLB (0.42) TSHRSSTR1SSTR4KMT2ADPP4
SCHEMBL23532545 0.66 TSHR (0.50) L3MBTL1TDP1ALDH1A1ECE1TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1912994-A1 ADENINE DERIVATIVES Merck Patent GmbH (DE) 2008-04-23 EP disclosed
WO-2007017069-A1 ADENINE DERIVATIVES MERCK PATENT GMBH (DE) 2007-02-15 WO disclosed