SCHEMBL4604495

SCHEMBL4604495

O=C(O)[C@H]1Cc2ccccc2CN1C(=O)Nc1ccc(Cl)cn1

nearest known ligand 0.59

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
F10 P00742 1/20 0.59
L3MBTL1 Q9Y468 3/20 0.54
TDP1 Q9NUW8 2/20 0.54
NAMPT P43490 1/20 0.52
POLB P06746 3/20 0.50
CYP3A4 P08684 1/20 0.46
CYP2C19 P33261 1/20 0.46
LMNA P02545 2/20 0.45
GAA P10253 1/20 0.45
ALDH1A1 P00352 1/20 0.45
NPSR1 Q6W5P4 2/20 0.45
MEN1 O00255 1/20 0.45
KMT2A Q03164 1/20 0.45
RAB9A P51151 4/20 0.44
NPC1 O15118 3/20 0.44
HTT P42858 2/20 0.44
ALOX15 P16050 1/20 0.44
ACE P12821 2/20 0.44
TSHR P16473 1/20 0.44
STAT1 P42224 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4558064 0.82 TAS1R3 (0.60) L3MBTL1TDP1POLBCYP3A4CYP2C19
SCHEMBL27431292 0.78 NPC1 (0.55) L3MBTL1TDP1POLBCYP3A4CYP2C19
SCHEMBL3830412 0.76 LMNA (0.56) L3MBTL1LMNAGAAALDH1A1KMT2A
SCHEMBL4606285 0.75 F10 (1.00) F10
SCHEMBL23657718 0.74 NPY5R (0.57) L3MBTL1TDP1NAMPTLMNAGAA
SCHEMBL4111979 0.73 TDP1 (0.62) L3MBTL1TDP1POLBLMNAGAA
SCHEMBL11350319 0.73 ACE (0.59) L3MBTL1TDP1POLBLMNAALDH1A1
SCHEMBL3840630 0.71 ACE (0.61) L3MBTL1TDP1POLBLMNAALDH1A1
SCHEMBL4573235 0.71 ACE (0.61) L3MBTL1TDP1POLBLMNAALDH1A1
SCHEMBL8908771 0.71 ACE (0.61) L3MBTL1TDP1POLBLMNAALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1948639-A2 NOVEL CARBOCYCLIC FUSED CYCLIC AMINES F. Hoffmann-la Roche AG (CH) 2008-07-30 EP claimed
WO-2007054453-A2 CARBOCYCLIC FUSED CYCLIC AMINES AS INHIBITORS OF THE COAGULATION FACTOR XA F. HOFFMANN-LA ROCHE AG (CH) 2007-05-18 WO claimed