SCHEMBL4604943

SCHEMBL4604943

Cc1cc(-c2ccc(Cl)cc2)c(Cl)cc1Cl

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AHR P35869 5/20 0.47
HSD11B1 P28845 2/20 0.43
CD44 P16070 1/20 0.38
MEN1 O00255 1/20 0.38
NPC1 O15118 1/20 0.38
CYP1A2 P05177 1/20 0.38
CYP2C19 P33261 1/20 0.38
RAB9A P51151 1/20 0.38
KMT2A Q03164 1/20 0.38
SMN1; SMN2 Q16637 1/20 0.38
TDO2 P48775 1/20 0.37
KDM4E B2RXH2 1/20 0.37
ALDH1A1 P00352 1/20 0.37
HPGD P15428 1/20 0.37
PPARG P37231 1/20 0.37
STAT3 P40763 1/20 0.37
NPSR1 Q6W5P4 1/20 0.37
RXFP1 Q9HBX9 1/20 0.37
NR2E3 Q9Y5X4 1/20 0.37
NCOR2 Q9Y618 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10066082 0.87 AHR (0.45) AHRCD44MEN1NPC1CYP1A2
SCHEMBL29801189 0.81 AHR (0.65) AHRHSD11B1MEN1CYP1A2KMT2A
SCHEMBL4449938 0.81 AHR (0.65) AHRHSD11B1MEN1CYP1A2KMT2A
SCHEMBL18618154 0.79 ALDH1A1 (0.50) AHRMEN1CYP1A2CYP2C19KMT2A
SCHEMBL6452021 0.74 AHR (0.47) AHRHSD11B1CYP1A2PTGS2
SCHEMBL13906326 0.74 HSD11B1 (0.47) AHRHSD11B1MEN1NPC1RAB9A
Sulfur Dioxide SCHEMBL28329775 0.74 AHR (0.56) AHRHSD11B1MEN1CYP1A2KMT2A
SCHEMBL12054920 0.73 AHR (0.60) AHRMEN1CYP2C19KMT2AKDM4E
SCHEMBL680179 0.73 NOTUM (0.47) AHRHSD11B1CYP1A2CYP2C19PTGS2
SCHEMBL30487478 0.73 NOTUM (0.47) AHRHSD11B1CYP1A2CYP2C19PTGS2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1947090-A1 Method for preparing N-piperidino-1,5-diphenylpyrazole-3-carboxamide and derivatives Laboratorios del Dr. Esteve S.A. (ES) 2008-07-23 EP disclosed