SCHEMBL4607597

SCHEMBL4607597

O=C(O)NCCC(O)c1ccccc1F

nearest known ligand 0.54

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
CNR2 P34972 3/20 0.44
CES2 O00748 1/20 0.42
CES1 P23141 1/20 0.42
GAA P10253 1/20 0.42
MTNR1A P48039 1/20 0.39
MTNR1B P49286 1/20 0.39
NPC1 O15118 2/20 0.39
RAB9A P51151 2/20 0.39
PRMT3 O60678 1/20 0.39
CNR1 P21554 2/20 0.38
EPHX2 P34913 1/20 0.38
HIF1A Q16665 1/20 0.37
EEF2K O00418 1/20 0.37
MC4R P32245 1/20 0.37
CYP3A4 P08684 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL26907022 0.83 PRMT3 (0.48) CNR2CES2CES1GAANPC1
Hydrochloric Acid SCHEMBL382716 0.81 GAA (0.43) CNR2CES2CES1GAAMTNR1A
SCHEMBL14691232 0.79 CFD (0.40)
SCHEMBL13997820 0.79 MALT1 (0.45) GAAMC4R
SCHEMBL20213832 0.78 TAAR1 (0.46) CES2CES1CYP3A4
SCHEMBL11495829 0.78 CES2 (0.46) CNR2CES2CES1GAAEEF2K
SCHEMBL3510106 0.78 MTNR1A (0.53) CNR2MTNR1AMTNR1BNPC1RAB9A
SCHEMBL20580058 0.77 GAA (0.42) CNR2CES2CES1GAAPRMT3
SCHEMBL16371920 0.77 CES2 (0.43) CNR2CES2CES1GAACYP3A4
SCHEMBL5061358 0.76 POLB (0.43) NPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1874768-A2 INHIBITORS OF AKT ACTIVITY SMITHKLINE BEECHAM CORPORATION (US) 2008-01-09 EP disclosed
WO-2006113837-A2 INHIBITORS OF AKT ACTIVITY SMITHKLINE BEECHAM CORPORATION (US) 2006-10-26 WO disclosed