SCHEMBL4608265

SCHEMBL4608265

COC(=O)Oc1ccc2c(c1)NC(=O)N(C1CCN(Cc3ccccc3)CC1)C2

nearest known ligand 0.55

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
CHRM4 P08173 1/20 0.55
CHRM3 P20309 5/20 0.48
CHRM2 P08172 4/20 0.46
RAMP1 O60894 2/20 0.46
CALCRL Q16602 2/20 0.46
SIGMAR1 Q99720 2/20 0.45
CTSS P25774 3/20 0.44
DRD2 P14416 1/20 0.43
DRD4 P21917 1/20 0.43
MAOB P27338 1/20 0.43
CALCA P06881 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5091174 0.88 CHRM3 (0.58) CHRM4CHRM3CHRM2SIGMAR1DRD2
SCHEMBL3958065 0.85 CHRM4 (0.56) CHRM4CHRM3CHRM2RAMP1CALCRL
SCHEMBL5088985 0.81 CHRM4 (0.58) CHRM4CHRM3CHRM2RAMP1CALCRL
SCHEMBL4607869 0.81 MAPK1 (0.43) CHRM4RAMP1CALCRLCALCA
SCHEMBL2980917 0.79 CTSS (0.57) CHRM4CHRM3CHRM2CALCRLSIGMAR1
SCHEMBL9046543 0.78 CHRM4 (0.70) CHRM4CHRM3CHRM2RAMP1CALCRL
SCHEMBL3596998 0.75 CHRM4 (0.58) CHRM4CHRM3CHRM2RAMP1CALCRL
SCHEMBL3967246 0.75 CHRM4 (0.65) CHRM4CHRM3CHRM2RAMP1CALCRL
SCHEMBL8126590 0.74 OPRK1 (0.54) CHRM3CHRM2SIGMAR1DRD4
SCHEMBL2262403 0.74 CHRM3 (0.57) CHRM3CHRM2SIGMAR1DRD2DRD4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1440976-B1 Modified aminoacids, pharmaceuticals containing these compounds and method for their production BOEHRINGER INGELHEIM PHARMA (DE) 2008-07-23 EP disclosed
EP-1440976-A1 Modified aminoacids, pharmaceuticals containing these compounds and method for their production Boehringer Ingelheim Pharma GmbH & Co.KG (DE) 2004-07-28 EP disclosed
EP-0927192-B1 MODIFIED AMINOACIDS, PHARMACEUTICALS CONTAINING THESE COMPOUNDS AND METHOD FOR THEIR PRODUCTION BOEHRINGER INGELHEIM PHARMA (DE) 2004-05-12 EP disclosed