SCHEMBL460986

SCHEMBL460986

Brc1cnn2c(I)cnc2c1Br

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ABL1 P00519 1/20 0.38
KDR P35968 1/20 0.38
AXL P30530 1/20 0.32
PRKAB2 O43741 1/20 0.30
PRKAG1 P54619 1/20 0.30
PRKAA2 P54646 1/20 0.30
PRKAA1 Q13131 1/20 0.30
PRKAG3 Q9UGI9 1/20 0.30
PRKAG2 Q9UGJ0 1/20 0.30
PRKAB1 Q9Y478 1/20 0.30
NPC1 O15118 1/20 0.30
ALDH1A1 P00352 1/20 0.30
LMNA P02545 1/20 0.30
MAPT P10636 1/20 0.30
HTT P42858 1/20 0.30
RAB9A P51151 1/20 0.30
PAX8 Q06710 1/20 0.30
SMN1; SMN2 Q16637 1/20 0.30
NPSR1 Q6W5P4 1/20 0.30
RXFP1 Q9HBX9 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL457469 0.67 ABL1 (0.30) ABL1KDR
SCHEMBL23679750 0.64 PI4KA (0.35) ALDH1A1
SCHEMBL23104591 0.62 KDM4D (0.41) ABL1KDRALDH1A1LMNAHTT
SCHEMBL10176568 0.58
SCHEMBL24508317 0.58
SCHEMBL25332231 0.57 TRPA1 (0.34)
SCHEMBL23104263 0.56 GABRA1 (0.39)
SCHEMBL19336865 0.55 KDM4E (0.43) LMNAMAPTHTT
SCHEMBL3754835 0.54 PRKAB2 (0.54) ABL1KDRAXLPRKAB2PRKAG1
SCHEMBL867287 0.54 KDR (0.42) ABL1KDRAXLALDH1A1LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2614063-A1 SUBSTITUTED IMIDAZOPYRIDAZINES Bayer Intellectual Property GmbH (DE) 2013-07-17 EP disclosed
WO-2012032031-A1 SUBSTITUTED IMIDAZOPYRIDAZINES BAYER PHARMA AKTIENGESELLSCHAFT (DE) 2012-03-15 WO disclosed