SCHEMBL4610033

SCHEMBL4610033

O=C(O)N1CCC(N2C(=O)N(CC3OCCO3)CC2c2cccc(Cl)c2)CC1

nearest known ligand 0.43

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
CCR5 P51681 17/20 0.43
CCR4 P51679 1/20 0.42
KCNH2 Q12809 1/20 0.42
HDAC1 Q13547 1/20 0.42
HDAC6 Q9UBN7 1/20 0.42
HSD11B1 P28845 1/20 0.38
NPC1 O15118 1/20 0.38
KMT2A Q03164 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5573793 0.87 SMN1; SMN2 (0.44) CCR5CCR4KCNH2HDAC1HDAC6
SCHEMBL5576527 0.85 DRD2 (0.41) CCR5CCR4KCNH2HDAC1HDAC6
SCHEMBL4597857 0.78 CCR5 (0.57) CCR5CCR4KCNH2
SCHEMBL5575918 0.76 CCR5 (0.77) CCR5CCR4KCNH2
SCHEMBL4597655 0.75 CCR5 (0.43) CCR5CCR4KCNH2HDAC1HDAC6
SCHEMBL5575518 0.72 CCR5 (0.66) CCR5CCR4KCNH2
SCHEMBL4607778 0.71 DRD2 (0.44) CCR5CCR4KCNH2HDAC1HDAC6
SCHEMBL4595920 0.71 STS (0.44) CCR5HDAC1HDAC6KMT2A
SCHEMBL5576431 0.70 CCR5 (0.65) CCR5CCR4KCNH2
SCHEMBL4598523 0.68 CCR5 (0.60) CCR5CCR4KCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1924265-A2 CHEMOKINE RECEPTOR BINDING COMPOUNDS Genzyme Corporation (US) 2008-05-28 EP disclosed
WO-2007022371-A2 CHEMOKINE RECEPTOR BINDING COMPOUNDS GENZYME CORPORATION (US) 2007-02-22 WO disclosed