SCHEMBL4611702

SCHEMBL4611702

CCS(=O)(=O)c1ccc(CC(N)=O)cc1CN

nearest known ligand 0.41

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
PSIP1 O75475 1/20 0.41
CA2 P00918 1/20 0.40
KDM4E B2RXH2 2/20 0.39
LMNA P02545 1/20 0.39
POLB P06746 1/20 0.39
MAPK1 P28482 1/20 0.39
DDR1 Q08345 2/20 0.36
HTR2A P28223 1/20 0.36
SLC6A4 P31645 1/20 0.36
ALDH1A1 P00352 2/20 0.36
BACE1 P56817 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27993121 0.84 PSIP1 (0.53) PSIP1CA2KDM4EDDR1BACE1
SCHEMBL15358096 0.77 PSIP1 (0.40) PSIP1CA2LMNADDR1SLC6A4
Trifluoroacetic Acid SCHEMBL4613399 0.77 DDR1 (0.40) DDR1
Hydrochloric Acid SCHEMBL1017372 0.76 PSIP1 (0.39) PSIP1CA2LMNADDR1SLC6A4
SCHEMBL2853707 0.74 GAA (0.46) PSIP1CA2KDM4EMAPK1DDR1
SCHEMBL4683962 0.73 CA2 (0.50) CA2KDM4ELMNAPOLBMAPK1
SCHEMBL12997839 0.72 DDR1 (0.54) DDR1
SCHEMBL28247232 0.72 MMP2 (0.41) PSIP1CA2ALDH1A1
SCHEMBL27495350 0.72 CA2 (0.46) CA2KDM4ELMNAPOLBMAPK1
SCHEMBL16541866 0.72 DDR1 (0.44) PSIP1DDR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1910298-A2 PHENYLGLYCINAMIDE AND PYRIDYLGLYCINAMIDE DERIVATIVES USEFUL AS ANTICOAGULANTS Brystol-Myers Squibb Company (US) 2008-04-16 EP disclosed
WO-2007002313-A2 PHENYLGLYCINAMIDE AND PYRIDYLGLYCINAMIDE DERIVATIVES USEFUL AS ANTICOAGULANTS BRISTOL-MYERS SQUIBB COMPANY (US) 2007-01-04 WO disclosed